1. Signaling Pathways
  2. Vitamin D Related/Nuclear Receptor
  3. Estrogen Receptor/ERR
  4. Estrogen Receptor/ERR Inhibitors

Estrogen Receptor/ERR Inhibitors

Estrogen receptor

ERα

ERβ

ERRα

ERRβ

ERRγ

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Estrogen Receptor/ERR Degraders, Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name Estrogen receptor ERα ERβ ERRα ERRβ ERRγ Purity
Tamoxifen
Estrogen receptor
          99.92%
4-Hydroxytamoxifen
Estrogen receptor, IC50: 3.3 nM
          99.96%
Kaempferol  
ERα
        99.86%
Tamoxifen Citrate
Estrogen receptor
          99.95%
Propyl pyrazole triol  
ERα
        99.11%
DPN    
ERβ, EC50: 0.85 nM
      99.66%
XCT790      
ERRα, IC50: 0.37 μM
    99.54%
Saikosaponin D    
ERβ
      98.76%
Giredestrant
ER
          99.52%
(E/Z)-4-Hydroxytamoxifen
Estrogen receptor
          99.60%
DY131        
ERRβ
ERRγ
99.88%
GSK5182          
ERRγ, IC50: 79 nM
99.85%
Prinaberel  
hERα, IC50: 1200 nM
mouse ERα, IC50: 750 nM
rat ERα, IC50: 620 nM
hERβ, IC50: 5.4 nM
rat ERβ, IC50: 3.1 nM
mouse ERβ, IC50: 3.7 nM
      98.05%
ERRα antagonist-1      
ERRα
    98.48%
Amcenestrant  
ERα, EC50: 0.2 nM
        99.59%
SLU-PP-332      
ERRα, EC50: 98 nM
ERRβ, EC50: 230 nM
ERRγ, EC50: 430 nM
99.44%
Smurf1-IN-A01  
ERα
        99.90%
MPP dihydrochloride  
ERα
ERβ
      99.06%
DS45500853      
ERRα
    98.15%
PROTAC ERRα Degrader-3      
ERRα
    98.82%
Hexestrol  
ERα, Ki: 0.06 nM
ERβ, Ki: 0.06 nM
      99.89%
Tamoxifen (Standard)
Estrogen receptor
          99.76%
H3B-5942  
ERαY537S, Ki: 0.41 nM
ERαWT, Ki: 1 nM
        99.73%
Erteberel    
ERβ, Ki: 1.54 nM
ERβ, EC50: 3.61 nM
      99.87%
Raloxifene
Estrogen receptor
          99.62%
FLTX1  
ERα, IC50: 87.5 nM
        99.78%
PROTAC ERRα ligand 1      
ERRα, IC50: 0.04 μM
 
ERRγ, IC50: 2.8 μM
98.12%
GNE-149  
ERα, IC50: 0.053 nM
        99.66%
Acolbifene  
ERα, IC50: 2 nM (E2-induced transcriptional activity)
ERβ, IC50: 0.4 nM (E2-induced transcriptional activity)
      99.52%
Zearalanone
Estrogen receptor
          99.78%
ERRγ agonist-1          
ERRγ
98.70%
OP-1074  
ERα
ERβ
      99.47%
Acolbifene hydrochloride  
ERα, IC50: 2 nM (E2-induced transcriptional activity)
ERβ, IC50: 0.4 nM (E2-induced transcriptional activity)
      99.00%
DS20362725      
ERRα
    98.15%
PROTAC ERα Degrader-2  
ERα
        98.88%
(E)-4-Hydroxytamoxifen
Estrogen receptor
          98.27%
MPP hydrochloride  
ERα
ERβ
      99.58%
Estrogen receptor β antagonist 2  
ERα, IC50: 109.10 μM
ERβ, IC50: 0.63 μM
      98.39%
Ferutinin  
ERα, IC50: 33.1 nM
ERβ, IC50: 180.5 nM
      ≥99.0%
Tamoxifen-d5
Estrogen receptor
          99.99%
PROTAC ER Degrader-4
ER
          98.22%
ERα degrader-2  
ERα, IC50: 4.6 nM
        99.71%
Endoxifen  
ERα
        99.42%
Y134  
ERα, Ki: 0.09 nM
ERβ, Ki: 11.31 nM
     
(R,R)-THC  
ERα, Ki: 9.0 nM
ERβ, Ki: 3.6 nM
      ≥99.0%
ERRγ inverse agonist 1  
ERα, IC50: 1.240 μM
   
ERRβ, IC50: 1.330 μM
ERRγ, IC50: 0.040 μM
Giredestrant tartrate
Estrogen receptor
         
PROTAC ERRα Degrader-1      
ERRα
   
ERα degrader 5  
ERα, EC50: 1.1 nM
ERα, IC50: 0.9 nM
ERβ, IC50: 2.3 nM
     
4',2-Dihydroxy-4,6-dimethoxydihydrochalcone
Estrogen receptor
         
ERα antagonist 1  
ERα
       
FERb 033    
ERβ, EC50: 4.8 nM
ERβ, Ki: 7.1 nM
     
Kaempferol (Standard)  
ERα
       
Estrogen receptor antagonist 8
Estrogen receptor
         
AC-186  
ERα, EC50: 5000 nM
ERβ, EC50: 6 nM
     
PROTAC ERα Degrader-4  
ERα, Ki: 5.08 μM
ERβ, Ki: 26.20 μM
     
PROTAC ERα Degrader-6  
ERα, DC50: 0.12 μM
       
(±)-8-Prenylnaringenin  
ERα, IC50: 57 nM
ERβ, IC50: 68 nM
     
CMP8  
MGERα, IC50: 29 nM
MGRERα, IC50: 41 nM
hERα, IC50: 1100 nM
hERβ, IC50: 2200 nM
     
LX-039
Estrogen receptor, EC50: 2.29 nM
         
ER degrader 6  
ERα
       
ERRα antagonist-2      
ERRα, IC50: 0.80 μM
   
SR19881        
ERRβ, EC50: 0.63 μM
ERRγ, EC50: 0.39 μM
(+)-Medicarpin    
ERβ
     
ERRγ inverse agonist 2          
ERRγ, Kd: 6.5 μM
LY117018
Estrogen receptor
         
7β-Hydroxy-epi-androsterone    
ERβ
     
(1S,3R)-GNE-502  
ERα, EC50: 13 nM
       
Estrogen receptor-IN-1  
ERα, IC50: 13 μM
ERβ, IC50: 5 μM
     
PSDalpha  
ERα
       
Estrogen receptor modulator 6  
ERα, Ki: 8.4 nM
ERβ, Ki: 0.44 nM
     
LSD1/ER-IN-1  
ERα
ERβ
     
2-Hydroxyestrone
Estrogen receptor