1. Signaling Pathways
  2. Others
  3. Estrogen Receptor/ERR
  4. ERα Inhibitors

ERα Inhibitors

Estrogen receptor

ERα

ERβ

ERRα

ERRβ

ERRγ

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform ERα together.

Please try each isoform separately.

ERα Specific Inhibitors, Agonists & Antagonists
Product Name ERα ERβ ERRβ ERRγ ERα Selectivity Purity
SAR439859
ERα, EC50: 0.2 nM
      Selective Antagonist 99.25%
Propyl pyrazole triol
ERα
      Selective Agonist ≥99.0%
PROTAC ERα Degrader-2
ERα
      Selective Inhibitor 98.02%
H3B-5942
ERαY537S, Ki: 0.41 nM
ERαWT, Ki: 1 nM
      Selective Inhibitor 99.31%
Endoxifen
ERα
      Selective
FLTX1
ERα, IC50: 87.5 nM
      Selective Inhibitor
ERRγ Inverse Agonist 1
ERα, IC50: 1.240 μM
 
ERRβ, IC50: 1.330 μM
ERRγ, IC50: 0.040 μM
Selective Antagonist
CMP8
MGERα, IC50: 29 nM
MGRERα, IC50: 41 nM
hERα, IC50: 1100 nM
hERβ, IC50: 2200 nM
    Selective
Prinaberel
hERα, IC50: 1200 nM
mouse ERα, IC50: 750 nM
rat ERα, IC50: 620 nM
hERβ, IC50: 5.4 nM
rat ERβ, IC50: 3.1 nM
mouse ERβ, IC50: 3.7 nM
    Pan Agonist 98.62%
Hexestrol
ERα, Ki: 0.06 nM
ERβ, Ki: 0.06 nM
    Pan Agonist ≥98.0%
OP-1074
ERα
ERβ
    Pan Inhibitor
Kaempferol
ERα
      Inhibitor 99.62%