2. Metabolic Enzyme/Protease
  3. Phosphodiesterase (PDE)
  4. Enpp-1-IN-13

Enpp-1-IN-13 (Compound 1a) is an ectonucleotide pyrophosphatase/phosphodiesterase (ENPP) inhibitor with IC50 values of 1.29 μM and 20.2 μM against ENPP1 and ENPP3, respectively. Enpp-1-IN-13 shows anticancer activity.

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Enpp-1-IN-13

Enpp-1-IN-13 Estructura química

No. CAS : 2417022-19-4

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Enpp-1-IN-13 Related Antibodies

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PDE1 PDE2 PDE3 PDE4 PDE5 PDE6 PDE7 PDE9 PDE10 PDE11 PDE12 PDE8 Autotaxin

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Descripciòn

Enpp-1-IN-13 (Compound 1a) is an ectonucleotide pyrophosphatase/phosphodiesterase (ENPP) inhibitor with IC50 values of 1.29 μM and 20.2 μM against ENPP1 and ENPP3, respectively. Enpp-1-IN-13 shows anticancer activity[1].

IC50 & Target

IC50: 1.29 μM (ENPP1), 20.2 μM (ENPP3)[1]
In Vitro

Enpp-1-IN-13 (Compound 1a) (100 μM) shows cytotoxic effect with inhibition of 23.0 ± 2.2%, 35.1 ± 0.8% and 30.4 ± 0.1% against HeLa, MCF-7 and 1321N1 cells, respectively[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Enpp-1-IN-13 Related Antibodies
Peso molecular

512.03

Fòrmula

C28H22ClN5OS
No. CAS
SMILES

S=C(NC1=CC=CC=C1)NC2=CC=CC(N3N=C(C4=CC=C(OC)C(Cl)=C4)C(C5=CC=NC=C5)=C3)=C2
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
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Enpp-1-IN-13 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Enpp-1-IN-132417022-19-4Phosphodiesterase (PDE)anticancerHeLaMCF-71321N1Inhibitorinhibitorinhibit

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Nombre del producto:
Enpp-1-IN-13
Cat. No.:
HY-147998
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