2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. Lavoltidine

Lavoltidine  (Synonyms: Loxtidine; AH-234844)

製品番号: HY-121450
取扱説明書 Technical Support

Lavoltidine (Loxtidine) is an an orally active, irreversible and highly potent histamine H2-receptor antagonist. Lavoltidine strongly inhibits gastric acid secretion and also induces hypergastrinemia.

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Lavoltidine

Lavoltidine 構造式

CAS 番号 : 76956-02-0

容量 価格（税別） 在庫状況 数量
1 mg $544 お問い合わせ 2 - 3 weeks 1-2 weeks 3 - 4 weeks 2-3 weeks
5 mg $1353 お問い合わせ 2 - 3 weeks 1-2 weeks 3 - 4 weeks 2-3 weeks
10 mg $1960 お問い合わせ 2 - 3 weeks 1-2 weeks 3 - 4 weeks 2-3 weeks
25 mg $2915 お問い合わせ 2 - 3 weeks 1-2 weeks 3 - 4 weeks 2-3 weeks
50 mg $3905 お問い合わせ 2 - 3 weeks 1-2 weeks 3 - 4 weeks 2-3 weeks
100 mg $5280 お問い合わせ 2 - 3 weeks 1-2 weeks 3 - 4 weeks 2-3 weeks
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500 mg   お問い合わせ  
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Lavoltidine 関連抗体

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製品説明

Lavoltidine (Loxtidine) is an an orally active, irreversible and highly potent histamine H2-receptor antagonist. Lavoltidine strongly inhibits gastric acid secretion and also induces hypergastrinemia[1].

IC50 & Target

H2 Receptor

 

体内実験

Lavoltidine (Loxtidine; 0.5 g/L; orally (drinking water); changed weekly; for 3 months) shows partial suppression of both gastric acid secretion and progression to neoplasia. Lavoltidine inhibits gastric atrophy, hyperplasia, and dysplasia in H felis-infected INS-GAS mice[1].
Lavoltidine treatment for 6 months inhibits gastric tumors in H felis-infected INS-GAS mice[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male hypergastrinemic mice (INS-GAS mice) infected with Helicobacter felis[1]
Dosage: 0.5 g/L
Administration: Orally (drinking water); changed weekly; for 3 months
Result: Showed partial suppression of both gastric acid secretion and progression to neoplasia.
臨床実験
分子量

359.47

分子式

C19H29N5O2
CAS 番号
SMILES

OCC1=NN(C(NCCCOC2=CC=CC(CN3CCCCC3)=C2)=N1)C
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.
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参考文献
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Lavoltidine Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Lavoltidine76956-02-0Loxtidine AH-234844AH234844AH 234844AH-234844Histamine ReceptororallyirreversiblegastricacidsecretionhypergastrinemiatumorsHfelisInhibitorinhibitorinhibit

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製品名:
Lavoltidine
製品番号:
HY-121450
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