1. Signaling Pathways
  2. GPCR/G Protein
  3. Leukotriene Receptor
  4. Leukotriene Receptor Inhibitors

Leukotriene Receptor Inhibitors

LTB4

LTC4

LTD4/CysLT1

LTE4

CysLT2

CysLT1

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Leukotriene Receptor Inhibitors & Antagonists
Product Name LTB4 LTC4 LTD4/CysLT1 LTE4 CysLT2 CysLT1 Purity
Montelukast sodium          
CysLT1
99.52%
MK-571 sodium salt    
LTD4, Ki: 0.22 nM (In guinea pig lung)
LTD4, Ki: 2.1 nM (In human lung)
      99.24%
Zafirlukast    
LTD4
      99.90%
Fiboflapon
LTB4, IC50: 76 nM
          98.18%
Montelukast          
CysLT1
Pranlukast  
LTC4, Ki: 5640 nM
LTD4, Ki: 0.99 nM
LTE4, Ki: 0.63 nM
    99.98%
Gemilukast        
CysLT2, IC50: 25 nM (in human)
CysLT1, IC50: 1.7 nM (in human)
99.58%
Nedocromil  
LTC4
        98.86%
Pranlukast hemihydrate  
LTC4, Ki: 5640 nM
LTD4, Ki: 0.99 nM
LTE4, Ki: 0.63 nM
    99.93%
LY223982
LTB4, IC50: 13.2 nM
          >99.0%
Fiboflapon sodium
LTB4, IC50: 76 nM
          99.08%
Nedocromil sodium  
LTC4
       
Veliflapon
LTB4
LTC4
        >99.0%
Darbufelone mesylate
LTB4
         
DW-1350
LTB4
         
HAMI 3379        
CysLT2
  >95.0%
(S)-Verapamil hydrochloride  
LTC4
       
5-O-Demethylnobiletin  
LTC4, IC50: 0.35 μM
       
CP-105696
LTB4, IC50: 8.42±0.26 nM
         
LY255283
LTB4, IC50: ~100 nM (LTB4 binds to guinea pig lung membranes)
         
Amelubant
LTB4, Ki: 221 nM (in vital human granulocytes)
LTB4, Ki: 230 nM (in cell membranes)
         
CP-96021 hydrochloride  
LTC4, Ki: 34 nM
       
CP-96486    
LTD4, Ki: 20 nM
     
Quinotolast sodium  
LTC4
       
LM-1484  
LTC4
CysLT1
     
Tipelukast    
LTD4, pA2: 6.41 (In guinea-pigs)
LTE4, pA2: 6.45 (In guinea-pigs)
   
RS-601    
LTD4
     
ONO4057
LTB4, IC50: 0.7 μM
         
LTD4 antagonist 1    
LTD4, Ki: 0.57 nM
     
LY210073
LTB4, IC50: 6.2 nM
         
CI-949  
LTC4, IC50: 0.5 μM
LTD4, IC50: 0.5 μM
     
KP496    
LTD4
     
YM158 free base    
LTD4, pA2: 8.87
     
Bunaprolast
LTB4
         
LTB4-IN-1
LTB4, IC50: 70 nM