1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFR Inhibitors

PDGFR Inhibitors

PDGFR

PDGFRβ

PDGFRα

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PDGFR Inhibitors
Product Name PDGFR PDGFRβ PDGFRα Purity
Lenvatinib  
PDGFRβ, IC50: 39 nM
PDGFRα, IC50: 51 nM
99.87%
Nintedanib  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.97%
Regorafenib  
PDGFRβ, IC50: 22 nM
  ≥99.0%
Sunitinib  
PDGFRβ, IC50: 2 nM
  ≥98.0%
Dovitinib lactate hydrate  
PDGFRβ, IC50: 210 nM
PDGFRα, IC50: 27 nM
Chiauranib  
PDGFRβ, IC50: 93 nM
PDGFRα, IC50: 1 nM
99.28%
Ponatinib    
PDGFRα, IC50: 1.1 nM
99.13%
Axitinib  
PDGFRβ, IC50: 1.6 nM
  99.94%
Pazopanib  
PDGFRβ, IC50: 84 nM
  99.75%
SU 5402  
PDGFRβ, IC50: 510 nM
  99.39%
Crenolanib  
PDGFRβ, Kd: 3.2 nM
PDGFRα, Kd: 2.1 nM
99.67%
Sunitinib Malate  
PDGFRβ, IC50: 2 nM
  ≥99.0%
Nintedanib esylate  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.93%
Ripretinib    
PDGFRA
98.90%
Dovitinib  
PDGFRβ, IC50: 210 nM
PDGFRα, IC50: 27 nM
99.94%
Cediranib  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
≥98.0%
CP-673451  
PDGFRβ, IC50: 1 nM
PDGFRα, IC50: 10 nM
99.65%
Pazopanib Hydrochloride  
PDGFRβ, IC50: 84 nM
  99.84%
Amuvatinib    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
98.07%
Lenvatinib mesylate  
PDGFRβ, IC50: 39 nM
PDGFRα, IC50: 51 nM
99.86%
Linifanib  
PDGFRβ, IC50: 66 nM
  99.72%
ENMD-2076    
PDGFRα, IC50: 56.4 nM
99.12%
Regorafenib Hydrochloride  
PDGFRβ, IC50: 22 nM
  ≥98.0%
Telatinib    
PDGFRα, IC50: 15 nM
98.72%
CHIR-124
PDGFR, IC50: 6.6 nM
    ≥95.0%
Regorafenib monohydrate  
PDGFRβ, IC50: 22 nM
  99.96%
Ilorasertib hydrochloride  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
98.91%
TG 100801  
PDGFRβ, IC50: 13 nM
  ≥95.0%
Orantinib  
PDGFRβ, Ki: 8 nM
  98.80%
PP121
PDGFR, IC50: 2 nM
    99.08%
Tandutinib
PDGFR, IC50: 0.2 μM
    99.48%
SU14813  
PDGFRβ, IC50: 4 nM
  98.90%
Toceranib phosphate  
PDGFRβ, Ki: 5 nM
  98.02%
TAK-593  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
99.62%
PP58
PDGFR
    99.48%
Cediranib maleate  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
99.74%
Dovitinib lactate  
PDGFRβ, IC50: 210 nM
PDGFRα, IC50: 27 nM
99.96%
JI-101  
PDGFRβ
  99.95%
JNJ-10198409  
PDGFRβ, IC50: 4.2 nM
PDGFRα, IC50: 45 nM
≥99.0%
Toceranib  
PDGFRβ, Ki: 5 nM
  96.25%
Methylnissolin
PDGFR, IC50: 10 μM
    99.64%
SU16f
PDGFR2, IC50: 140 nM
PDGFR1, IC50: 2.29 μM
PDGFRβ, IC50: 10 nM
  ≥99.0%
AC710  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM
99.89%
Tandutinib hydrochloride
PDGFR, IC50: 0.2 μM
    98.84%
Tyrphostin AG1433  
PDGFRβ, IC50: 5 μM
  99.20%
Tyrphostin AG1296  
PDGFRβ
PDGFRα
99.25%
Tyrosine kinase-IN-1    
PDGFRα, IC50: 4 nM
99.47%
ENMD-2076 Tartrate    
PDGFRα, IC50: 56.4 nM
98.87%
SU14813 maleate  
PDGFRβ, IC50: 4 nM
  99.95%
AZD2932  
PDGFRβ, IC50: 4 nM
  ≥98.0%
PDGFRα kinase inhibitor 1  
PDGFRβ, IC50: 6115 nM
PDGFRα, IC50: 132 nM
99.90%
NVP-ACC789  
PDGFR-β, IC50: 1.4 μM
  99.94%
PD-161570
PDGFR, IC50: 310 nM
PDGFRβ, IC50: 262 nM
  99.04%
SU4312
PDGFR
    98.19%
(Z)-Orantinib  
PDGFRβ, IC50: 0.008 μM
  99.02%
Hypothemycin  
PDGFRβ, Ki: 900 nM
PDGFRα, Ki: 1.5 μM
≥98.0%
TG 100572  
PDGFRβ, IC50: 13 nM
 
Ilorasertib  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
≥98.0%
GZD856  
PDGFRβ, IC50: 136.6 nM
PDGFRα, IC50: 68.6 nM
Telatinib mesylate    
PDGFRα, IC50: 15 nM
Amuvatinib hydrochloride    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
GZD856 formic  
PDGFRβ, IC50: 136.6 nM
PDGFRα, IC50: 68.6 nM
98.06%
KG5  
PDGFRβ, Kd: 520 nM
PDGFRα, Kd: 300 nM
PD-089828  
PDGFR-β, IC50: 1.76 μM
PDGFR-β, Ki: 2.38 μM
 
Multi-kinase inhibitor 1
PDGFR
   
HG-7-85-01    
PDGFRα, IC50: 440 nM
Sunitinib D10  
PDGFRβ, IC50: 2 nM
 
Ponatinib D8    
PDGFRα, IC50: 1.1 nM
TG 100801 Hydrochloride  
PDGFRβ, IC50: 13 nM
 
AC710 Mesylate  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM