1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFR Inhibitors

PDGFR Inhibitors

PDGFR

PDGFRβ

PDGFRα

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PDGFR Inhibitors
Product Name PDGFR PDGFRβ PDGFRα Purity
Lenvatinib  
PDGFRβ, IC50: 39 nM
PDGFRα, IC50: 51 nM
99.74%
Nintedanib  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.97%
Regorafenib  
PDGFRβ, IC50: 22 nM
  99.96%
Sunitinib  
PDGFRβ, IC50: 2 nM
  99.66%
Ponatinib    
PDGFRα, IC50: 1.1 nM
99.13%
Tyrphostin AG1433  
PDGFRβ, IC50: 5 μM
  99.20%
Telatinib mesylate    
PDGFRα, IC50: 15 nM
Axitinib  
PDGFRβ, IC50: 1.6 nM
  99.94%
Crenolanib  
PDGFRβ, Kd: 3.2 nM
PDGFRα, Kd: 2.1 nM
99.67%
SU 5402  
PDGFRβ, IC50: 510 nM
  99.39%
Cediranib  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
99.58%
Ripretinib    
PDGFRA
99.46%
CP-673451  
PDGFRβ, IC50: 1 nM
PDGFRα, IC50: 10 nM
99.65%
Sunitinib Malate  
PDGFRβ, IC50: 2 nM
  99.47%
Nintedanib esylate  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.93%
Linifanib  
PDGFRβ, IC50: 66 nM
  99.60%
Dovitinib  
PDGFRβ, IC50: 210 nM
PDGFRα, IC50: 27 nM
97.18%
CHIR-124
PDGFR, IC50: 6.6 nM
    98.07%
SU14813  
PDGFRβ, IC50: 4 nM
  98.90%
Amuvatinib    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
99.36%
Pazopanib Hydrochloride  
PDGFRβ, IC50: 84 nM
  99.83%
Regorafenib Hydrochloride  
PDGFRβ, IC50: 22 nM
  99.58%
Regorafenib monohydrate  
PDGFRβ, IC50: 22 nM
  99.96%
PP121
PDGFR, IC50: 2 nM
    98.89%
ENMD-2076    
PDGFRα, IC50: 56.4 nM
99.23%
Tandutinib
PDGFR, IC50: 0.2 μM
    99.48%
Telatinib    
PDGFRα, IC50: 15 nM
99.49%
Ilorasertib hydrochloride  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
98.91%
Toceranib phosphate  
PDGFRβ, Ki: 5 nM
  98.43%
TAK-593  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
99.62%
ENMD-2076 Tartrate    
PDGFRα, IC50: 56.4 nM
98.59%
PP58
PDGFR
    98.94%
Orantinib  
PDGFRβ, Ki: 8 nM
  98.80%
Toceranib  
PDGFRβ, Ki: 5 nM
  96.25%
Cediranib maleate  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
96.67%
SU14813 maleate  
PDGFRβ, IC50: 4 nM
  99.95%
Tandutinib hydrochloride
PDGFR, IC50: 0.2 μM
    98.84%
AC710  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM
98.03%
NVP-ACC789  
PDGFR-β, IC50: 1.4 μM
  99.58%
JI-101  
PDGFRβ
  99.95%
JNJ-​10198409  
PDGFRβ, IC50: 4.2 nM
PDGFRα, IC50: 45 nM
>99.0%
PDGFRα kinase inhibitor 1  
PDGFRβ, IC50: 6115 nM
PDGFRα, IC50: 132 nM
99.90%
SU16f
PDGFR2, IC50: 140 nM
PDGFR1, IC50: 2.29 μM
PDGFRβ, IC50: 10 nM
  >99.0%
Tyrosine kinase-IN-1    
PDGFRα, IC50: 4 nM
99.47%
Ilorasertib  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
AZD2932  
PDGFRβ, IC50: 4 nM
  98.12%
Lenvatinib mesylate  
PDGFRβ, IC50: 39 nM
PDGFRα, IC50: 51 nM
GZD856  
PDGFRβ, IC50: 136.6 nM
PDGFRα, IC50: 68.6 nM
Amuvatinib hydrochloride    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
Methylnissolin
PDGFR, IC50: 10 μM
   
PD-089828  
PDGFR-β, IC50: 1.76 μM
PDGFR-β, Ki: 2.38 μM
 
Multi-kinase inhibitor 1
PDGFR
   
PD-161570
PDGFR, IC50: 310 nM
PDGFRβ, IC50: 262 nM
 
Hypothemycin  
PDGFRβ, Ki: 900 nM
PDGFRα, Ki: 1.5 μM
HG-7-85-01    
PDGFRα, IC50: 440 nM
Sunitinib D10  
PDGFRβ, IC50: 2 nM
 
Ponatinib D8    
PDGFRα, IC50: 1.1 nM
SKLB610
PDGFR
    99.23%
AC710 Mesylate  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM