1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. PDGFR
  4. PDGFR Inhibitors

PDGFR Inhibitors

PDGFR

PDGFRβ

PDGFRα

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PDGFR Inhibitors
Product Name PDGFR PDGFRβ PDGFRα Purity
Nintedanib  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.97%
Regorafenib  
PDGFRβ, IC50: 22 nM
  99.96%
Imatinib
PDGFR, IC50: 100 nM
    99.80%
PDGFRα kinase inhibitor 1  
PDGFRβ, IC50: 6115 nM
PDGFRα, IC50: 132 nM
Methylnissolin
PDGFR, IC50: 10 μM
   
Crenolanib  
PDGFRβ, Kd: 3.2 nM
PDGFRα, Kd: 2.1 nM
99.78%
Axitinib  
PDGFRβ, IC50: 1.6 nM
  99.94%
Sunitinib Malate  
PDGFRβ, IC50: 2 nM
  99.47%
SU 5402  
PDGFRβ, IC50: 510 nM
  99.39%
Cediranib  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
99.58%
CP-673451  
PDGFRβ, IC50: 1 nM
PDGFRα, IC50: 10 nM
99.65%
Nintedanib esylate  
PDGFRβ, IC50: 65 nM
PDGFRα, IC50: 59 nM
99.95%
Ripretinib    
PDGFRA
99.46%
CHIR-124
PDGFR, IC50: 6.6 nM
    98.77%
SU14813  
PDGFRβ, IC50: 4 nM
  95.74%
Regorafenib Hydrochloride  
PDGFRβ, IC50: 22 nM
  99.58%
Pazopanib Hydrochloride  
PDGFRβ, IC50: 84 nM
  99.92%
PP121
PDGFR, IC50: 2 nM
    98.89%
TAK-593  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 4.3 nM
PDGFRαV561D, IC50: 1 nM
99.62%
Regorafenib monohydrate  
PDGFRβ, IC50: 22 nM
  99.96%
Telatinib    
PDGFRα, IC50: 15 nM
99.49%
Amuvatinib    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
99.36%
Toceranib phosphate  
PDGFRβ, Ki: 5 nM
  98.43%
PP58
PDGFR
    98.07%
Toceranib  
PDGFRβ, Ki: 5 nM
  96.50%
SU14813 maleate  
PDGFRβ, IC50: 4 nM
  99.34%
Orantinib  
PDGFRβ, Ki: 0.008 μM
  99.02%
JI-101  
PDGFRβ
  99.95%
Cediranib maleate  
PDGFRβ, IC50: 5 nM
PDGFRα, IC50: 36 nM
96.67%
AC710  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM
98.03%
AZD2932  
PDGFRβ, IC50: 4 nM
  98.12%
NVP-ACC789  
PDGFR-β, IC50: 1.4 μM
  99.58%
Ilorasertib  
PDGFRβ, IC50: 13 nM
PDGFRα, IC50: 11 nM
Tyrosine kinase-IN-1    
PDGFRα, IC50: 4 nM
99.47%
GZD856  
PDGFRβ, IC50: 136.6 nM
PDGFRα, IC50: 68.6 nM
Amuvatinib hydrochloride    
PDGFRαV561D, IC50: 40 nM
PDGFRαD842V, IC50: 81 nM
SKLB610
PDGFR
    98.96%
AC710 Mesylate  
PDGFRβ, Kd: 1 nM
PDGFRα, Kd: 1.3 nM