1. Signaling Pathways
  2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine A2A receptor (A2AR) Inhibitors

Adenosine A2A receptor (A2AR) Inhibitors

Adenosine A1 receptor (A1R)

Adenosine A2A receptor (A2AR)

Adenosine A2B receptor (A2BR)

Adenosine A3 receptor (A3R)

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Sorry. There is currently no product that acts on isoform Adenosine A2A receptor (A2AR) together.

Please try each isoform separately.

Adenosine A2A receptor (A2AR) Specific Inhibitors & Antagonists
Product Name Adenosine A2A receptor (A2AR) Adenosine A1 receptor (A1R) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R) Adenosine A2A receptor (A2AR) Selectivity Purity
Adenosine receptor inhibitor 2
A2AR, Ki: 167 ± 22 nM
A1AR, Ki: 52.2 ± 8.5 nM
hA2B, Ki: >1000 nM
Adenosine A3 receptor, Ki: >1000 nM
Selective Inhibitor
ANR94
A2AR, Ki: 46 nM (human)
      Selective Antagonist
Adenosine receptor inhibitor 1
A2AR, Ki: 68.5 nM
A1AR, Ki: >1000 nM
hA2B, Ki: >1000 nM
Adenosine A3 receptor, Ki: >1000 nM
Selective Inhibitor
hA2A/hCA XII modulator 1
hA2AAR, Ki: 6.4 nM
hA1AR, Ki: 4.819 μM
 
hA3, Ki: >30 μM
Selective Antagonist
(E)-8-(3-Chlorostyryl)caffeine
A2AR
      Selective Antagonist
A2A receptor antagonist 2
A2AR, IC50: 8.3 nM
      Selective Antagonist
Adenosine receptor antagonist 1
A2AR, IC50: 0.29 nM
      Selective Antagonist
Adenosine receptor antagonist 2
A2a adenosine receptor, IC50: 1 nM
A2b adenosine receptor, IC50: 3 nM
      Pan Antagonist
A1AR antagonist 5
hA2AAR, pKi: <4
hA1AR, pKi: 6.11
    Pan Antagonist
A1AR antagonist 4
hA2AAR, pKi: <4
hA1AR, pKi: 6.29
    Pan Antagonist
MRS1334
rA2A, Ki: >100 nM
rA1, Ki: >100 nM
 
hA3, Ki: 2.69 nM
Pan Antagonist
A1AR antagonist 6
hA2AAR, pKi: <4
hA1AR, pKi: 7.13
    Pan Antagonist
PSB36
rA2A, Ki: 552 nM
rA1, Ki: 0.12 nM
hA2B, Ki: 187 nM
hA3, Ki: 2300 nM
rA3, Ki: 6500 nM
Pan Antagonist
A2A/A3 AR antagonist-1
hA2AAR, Ki: 90 nM
   
hA3, Ki: 31.8 nM
Pan Antagonist