1. GPCR/G Protein
  2. Adenosine Receptor
  3. LUF5834

LUF5834 is a selective A2B adenosine receptor (A2BR) partial agonist (EC50 = 12 nM). LUF5834 is also a partial A1/A2A adenosine receptor agonist (lacking selectivity) with Ki values of 2.6 and 28 nM, respectively.

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LUF5834 Chemical Structure

LUF5834 Chemical Structure

CAS No. : 333962-91-7

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Description

LUF5834 is a selective A2B adenosine receptor (A2BR) partial agonist (EC50 = 12 nM). LUF5834 is also a partial A1/A2A adenosine receptor agonist (lacking selectivity) with Ki values of 2.6 and 28 nM, respectively[1][2].

IC50 & Target[1]

A2BR

12 nM (EC50)

A2AR

28 nM (Ki)

A1R

2.6 nM (Ki)

Molecular Weight

348.38

Formula

C17H12N6OS

CAS No.
SMILES

N#CC1=C(C2=CC=C(O)C=C2)C(C#N)=C(SCC3=NC=CN3)N=C1N

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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LUF5834 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
LUF5834
Cat. No.:
HY-103170
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