1. Signaling Pathways
  2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine Receptor Inhibitors

Adenosine Receptor Inhibitors

Adenosine A1 receptor (A1R)

Adenosine A2A receptor (A2AR)

Adenosine A2B receptor (A2BR)

Adenosine A3 receptor (A3R)

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Adenosine Receptor Inhibitors, Agonists, Antagonists & Modulators
Product Name Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R) Purity
2'-MeCCPA
A1AR
      ≥98.0%
Derenofylline
A1R, Ki: 1 nM
A2AR, Ki: 398 nM
 
Adenosine A3 receptor, Ki: 200 nM
≥99.0%
MIPS521
A1AR
      99.65%
M1069  
A2AR
A2BR
 
Adenosine receptor antagonist 2  
A2a adenosine receptor, IC50: 1 nM
A2b adenosine receptor, IC50: 3 nM
    99.37%
Adenosine receptor inhibitor 2
A1AR, Ki: 52.2 ± 8.5 nM
A2AR, Ki: 167 ± 22 nM
hA2B, Ki: >1000 nM
Adenosine A3 receptor, Ki: >1000 nM
A1AR antagonist 5
hA1AR, pKi: 6.11
hA2AAR, pKi: <4
   
ANR94  
A2AR, Ki: 46 nM (human)
   
Adenosine receptor inhibitor 1
A1AR, Ki: >1000 nM
A2AR, Ki: 68.5 nM
hA2B, Ki: >1000 nM
Adenosine A3 receptor, Ki: >1000 nM
A1AR antagonist 4
hA1AR, pKi: 6.29
hA2AAR, pKi: <4
   
MRS1334
rA1, Ki: >100 nM
rA2A, Ki: >100 nM
 
hA3, Ki: 2.69 nM
hA3AR agonist 1      
Adenosine A3 receptor, Ki: 2.40 nM
LJ-4517  
A2AR, Ki: 18.3 nM
   
A1AR antagonist 6
hA1AR, pKi: 7.13
hA2AAR, pKi: <4
   
ISAM-140    
hA2B, Ki: 3.49 nM
 
A2A receptor antagonist 3
A1R, Ki: 107 nM
A2AR, Ki: 0.4 nM
A2BR, Ki: 37 nM
A3R, Ki: 1467 nM
hA2A/hCA XII modulator 1
hA1AR, Ki: 4.819 μM
hA2AAR, Ki: 6.4 nM
 
hA3, Ki: >30 μM
VCP171
A1R
     
A2AAR/HDAC-IN-1
A1AR, Ki: 503.3 ± 14 nM
A2AR, Ki: 163.5 ± 14 nM
hA2B, Ki: >10000 nM
Adenosine A3 receptor, Ki: >10000 nM
(E)-8-(3-Chlorostyryl)caffeine  
A2AR
   
Neladenoson dalanate hydrochloride
A1R
     
A2A receptor antagonist 2  
A2AR, IC50: 8.3 nM
   
VUF-5574      
Recombinant Human Adenosine A3 receptor (A3R) , Ki: 4.03 nM
A3AR antagonist 1      
hA3, Ki: 4.63 nM
PSB36
rA1, Ki: 0.12 nM
rA2A, Ki: 552 nM
hA2B, Ki: 187 nM
hA3, Ki: 2300 nM
rA3, Ki: 6500 nM
Neladenoson dalanate
A1R
     
MRS5698      
Adenosine A3 receptor, Ki: ~3 nM
A2A/A3 AR antagonist-1  
hA2AAR, Ki: 90 nM
 
hA3, Ki: 31.8 nM
A1AR antagonist 3
human A1, Ki: 9.69 nM
rat A1, Ki: 0.529 nM
     
A1/A3 AR antagonist 1
human A1, Ki: 36.7 nM
rat A1, Ki: 1.47 nM
   
human A3, Ki: 25.4 nM
Adenosine receptor antagonist 1  
A2AR, IC50: 0.29 nM