1. Signaling Pathways
  2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine A3 receptor (A3R) Inhibitors

Adenosine A3 receptor (A3R) Inhibitors

Adenosine A1 receptor (A1R)

Adenosine A2A receptor (A2AR)

Adenosine A2B receptor (A2BR)

Adenosine A3 receptor (A3R)

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Sorry. There is currently no product that acts on isoform Adenosine A3 receptor (A3R) together.

Please try each isoform separately.

Adenosine A3 receptor (A3R) Specific Inhibitors, Agonists & Antagonists
Product Name Adenosine A3 receptor (A3R) Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R) Selectivity Purity
MRS1334
hA3, Ki: 2.69 nM
rA1, Ki: >100 nM
rA2A, Ki: >100 nM
  Selective Antagonist
hA3AR agonist 1
Adenosine A3 receptor, Ki: 2.40 nM
      Selective Agonist
VUF-5574
Recombinant Human Adenosine A3 receptor (A3R) , Ki: 4.03 nM
      Selective Antagonist
A3AR antagonist 1
hA3, Ki: 4.63 nM
      Selective Antagonist
MRS5698
Adenosine A3 receptor, Ki: ~3 nM
      Selective Agonist
A1/A3 AR antagonist 1
human A3, Ki: 25.4 nM
human A1, Ki: 36.7 nM
rat A1, Ki: 1.47 nM
    Selective Antagonist
Adenosine receptor inhibitor 2
Adenosine A3 receptor, Ki: >1000 nM
A1AR, Ki: 52.2 ± 8.5 nM
A2AR, Ki: 167 ± 22 nM
hA2B, Ki: >1000 nM
Pan Inhibitor
Adenosine receptor inhibitor 1
Adenosine A3 receptor, Ki: >1000 nM
A1AR, Ki: >1000 nM
A2AR, Ki: 68.5 nM
hA2B, Ki: >1000 nM
Pan Inhibitor
hA2A/hCA XII modulator 1
hA3, Ki: >30 μM
hA1AR, Ki: 4.819 μM
hA2AAR, Ki: 6.4 nM
  Pan Antagonist
PSB36
hA3, Ki: 2300 nM
rA3, Ki: 6500 nM
rA1, Ki: 0.12 nM
rA2A, Ki: 552 nM
hA2B, Ki: 187 nM
Pan Antagonist
A2A/A3 AR antagonist-1
hA3, Ki: 31.8 nM
 
hA2AAR, Ki: 90 nM
  Pan Antagonist