Adenosine receptor antagonist 5
Adenosine receptor antagonist 5 (Compound 39) is a selective antagonist for human adenosine A3 receptor (hA3R) with Ki of 12 nM. Adenosine receptor antagonist 5 inhibits IB-MECA (HY-13591)-induced cAMP accumulation in NCI-H1792 cell, inhibits the proliferation of cancer cell LK-2 and NCI-H1792. Adenosine receptor antagonist 5 exhibits a fast metabolic rate in human liver microsomes.
For research use only. We do not sell to patients.
- Formula: C17H11BrCl2N4O3
- Molecular Weight:470.10
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Adenosine Receptor Isoforms
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Biological Activity
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human A3 12 nM (Ki) |
Chemical Information
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Molecular Weight 470.10
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Formula C17H11BrCl2N4O3
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SMILES
CC1=C(C(C2=C(C=CC=C2Cl)Cl)=NO1)C(O/N=C(C3=CC=C(C=N3)Br)\N)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Adenosine receptor antagonist 5 Related Classifications
HY-162787 Related Classifications
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