1. Signaling Pathways
  2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine A1 receptor (A1R) Inhibitors

Adenosine A1 receptor (A1R) Inhibitors

Adenosine A1 receptor (A1R)

Adenosine A2A receptor (A2AR)

Adenosine A2B receptor (A2BR)

Adenosine A3 receptor (A3R)

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform Adenosine A1 receptor (A1R) together.

Please try each isoform separately.

Adenosine A1 receptor (A1R) Specific Agonists & Antagonists
Product Name Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R) Adenosine A1 receptor (A1R) Selectivity Purity
MIPS521
A1AR
      Selective Agonist 99.65%
A1AR antagonist 5
hA1AR, pKi: 6.11
hA2AAR, pKi: <4
    Selective Antagonist
A1AR antagonist 4
hA1AR, pKi: 6.29
hA2AAR, pKi: <4
    Selective Antagonist
A1AR antagonist 6
hA1AR, pKi: 7.13
hA2AAR, pKi: <4
    Selective Antagonist
PSB36
rA1, Ki: 0.12 nM
rA2A, Ki: 552 nM
hA2B, Ki: 187 nM
hA3, Ki: 2300 nM
rA3, Ki: 6500 nM
Selective Antagonist
MRS1334
rA1, Ki: >100 nM
rA2A, Ki: >100 nM
 
hA3, Ki: 2.69 nM
Pan Antagonist
hA2A/hCA XII modulator 1
hA1AR, Ki: 4.819 μM
hA2AAR, Ki: 6.4 nM
 
hA3, Ki: >30 μM
Pan Antagonist