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Cat. No.: HY-139694

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hA3AR agonist 1

hA3AR agonist 1 is a potent human A₃ adenosine receptor (hA₃AR) agonist with a K_i value of 2.40 nM.

For research use only. We do not sell to patients.

CAS No.: 2821704-65-6
Formula: C₁₀H₁₄N₆OS
Molecular Weight:266.32

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

hA3AR agonist 1 Chemical Structure

CAS No.: 2821704-65-6

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
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Biological Activity

Description

hA3AR agonist 1 is a potent human A₃ adenosine receptor (hA₃AR) agonist with a K_i value of 2.40 nM.

IC₅₀ & Target

Adenosine A₃ receptor

2.40 nM (Ki)

All Adenosine Receptor Isoforms :

Chemical Information

CAS No. 2821704-65-6
Molecular Weight 266.32
Formula C₁₀H₁₄N₆OS
SMILES

O[C@H]1[C@H](N2C=NC3=C(NC)N=CN=C23)SC[C@H]1N
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Lee Y, et al. Subtle Chemical Changes Cross the Boundary between Agonist and Antagonist: New A3 Adenosine Receptor Homology Models and Structural Network Analysis Can Predict This Boundary. J Med Chem. 2021 Sep 9;64(17):12525-12536. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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hA3AR agonist 1

All Adenosine Receptor Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

hA3AR agonist 1 Related Classifications

HY-139694 Related Classifications