A3AR antagonist 3
A3AR antagonist 3 (compound 21) is a selective A3 adenosine receptor (A3AR) antagonist with a Ki of 37 nM. A3AR antagonist 3 shows >60-fold selectivity in comparison to A1 and A2A adenosine receptors.
For research use only. We do not sell to patients.
- CAS No.: 863202-33-9
- Formula: C17H18N6
- Molecular Weight:306.37
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adenosine Receptor Isoforms
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Biological Activity
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hA3 37 nM (Ki) |
hA1AR 2.22 μM (Ki) |
hA2AAR 7.73 μM (Ki) |
Chemical Information
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CAS No. 863202-33-9
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Molecular Weight 306.37
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Formula C17H18N6
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SMILES
[H][C@@]12[C@H]([C@@](C2)([H])CC1)NC3=C4N=CNC4=NC(NC5=CC=CC=C5)=N3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)