LUF5437
LUF5437 is a potent and selective adenosine A1 receptor antagonist with a rat Ki of 7.3 nM. LUF5437 can be used for research on cardiovascular and neurological diseases.
For research use only. We do not sell to patients.
- CAS No.: 331472-34-5
- Formula: C15H11N3O2S
- Molecular Weight:297.33
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adenosine Receptor Isoforms
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Biological Activity
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rA1 7.3 nM (Ki) |
rA2A 0.57 μM (Ki) |
hA3 0.13 μM (Ki) |
LUF5437 (Compound 8h) acts as a potent and selective adenosine A1 receptor antagonist, with a Ki of 7.3 nM at rat adenosine A1 receptors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 331472-34-5
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Molecular Weight 297.33
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Formula C15H11N3O2S
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SMILES
O=C(NC1=NC(C2=CC=CC=C2)=NS1)C3=CC=C(O)C=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)