1. Cell Cycle/DNA Damage
    Epigenetics
  2. PARP
  3. TNKS2/PARP5B Inhibitors

TNKS2/PARP5B Inhibitors

PARP

PARP1

PARP2

PARP3

PARP4

TNKS1/PARP5A

TNKS2/PARP5B

PARP10

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform TNKS2/PARP5B together.

Please try each isoform separately.

TNKS2/PARP5B Specific Inhibitors
Product Name TNKS2/PARP5B PARP1 PARP2 PARP3 TNKS1/PARP5A PARP10 TNKS2/PARP5B Selectivity Purity
NVP-TNKS656
TNKS2, IC50: 6 nM
 
PARP2, IC50: 32 μM
      Selective Inhibitor 99.14%
XAV-939
TNKS2, IC50: 2 nM
ARTD1, IC50: 5500 nM
ARTD2, IC50: 479 nM
 
TNKS1, IC50: 5 nM
  Pan Inhibitor 98.04%
RK-287107
tankyrase-2, IC50: 10.6 nM
     
tankyrase-1, IC50: 14.3 nM
  Pan Inhibitor
G007-LK
TNKS2, IC50: 25 nM
     
TNKS1, IC50: 46 nM
  Pan Inhibitor 99.24%
MN-64
TNKS2, IC50: 72 nM
ARTD1, IC50: 19.1 μM
ARTD2, IC50: 39.4 μM
 
TNKS1, IC50: 6 nM
  Pan Inhibitor 98.22%
ME0328
ARTD6/TNKS2, IC50: 34.3 μM
ARTD1/PARP1, IC50: 6.3 μM
ARTD2/PARP2, IC50: 10.8 μM
ARTD3/PARP3, IC50: 0.89 μM
ARTD5/TNKS1, IC50: 47.3 μM
ARTD10/PARP10, IC50: 71.3 μM
Pan Inhibitor 99.34%
K-756
TNKS2, IC50: 36 nM
     
TNKS1, IC50: 31 nM
  Pan Inhibitor >99.0%