1. Signaling Pathways
  2. GPCR/G Protein
  3. LPL Receptor
  4. LPL Receptor Inhibitors

LPL Receptor Inhibitors

LPAR1

LPAR2

LPAR3

LPAR5

S1PR1

S1PR3

S1PR4

S1PR5

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

LPL Receptor Inhibitors, Agonists & Antagonists
Product Name LPAR1 LPAR2 LPAR3 LPAR5 S1PR1 S1PR3 S1PR4 S1PR5 Purity
TAK-615
LPA1 Receptor, Kd: 1.7-14.5 nM
              99.51%
GRI977143  
LPA2 Receptor, EC50: 3.3 μM
           
Ponesimod        
S1PR1, IC50: 6 nM
S1PR3, IC50: 2068 nM
S1PR4, IC50: 1956 nM
S1PR5, IC50: 142 nM
99.72%
Cenerimod        
S1PR1, EC50: 1 nM
 
S1PR4, EC50: 2134 nM
S1PR5, EC50: 36 nM
S1PR5, EC50: 228 nM
≥98.0%
RP101075        
S1PR1, EC50: 0.27 nM
   
S1PR5, EC50: 5.9 nM
CYM50358            
S1PR4, IC50: 25 nM
 
NSC12404  
LPA2 Receptor
           
RP101442        
S1PR1, EC50: 2.6 nM
   
S1PR5, EC50: 171 nM
H2L 5765834
LPA1 Receptor, IC50: 94 nM
 
LPA3 Receptor, IC50: 752 nM
LPA5 Receptor, IC50: 463 nM