1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. ROR
  4. RORγ Inhibitors

RORγ Inhibitors

RORγ

RORα

RORβ

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform RORγ together.

Please try each isoform separately.

RORγ Specific Inhibitors & Antagonists
Product Name RORγ RORα RORβ RORγ Selectivity Purity
S18-000003
RORγt, IC50: <30 nM
    Selective Inhibitor
XY018
ROR-γ, IC50: 0.19 μM (in 293 T cells)
ROR-α, IC50: 7.57 μM (in 293 T cells)
  Selective Antagonist 99.76%
GNE-6468
ROR-γ, EC50: 2 nM
    Selective Antagonist 99.50%
Vimirogant hydrochloride
RORγt, Ki: 3.5 nM
RORγt, IC50: 17 nM
    Selective Inhibitor 98.33%
BMS-986251
RORγt, EC50: 12 nM
RORα, EC50: >10 μM
RORβ, EC50: >10 μM
Selective Antagonist
RORγt Inverse agonist 10
RORγt, IC50: 51 nM
    Selective Antagonist
A-9758
RORγt, IC50: 5 nM
    Selective Inhibitor
Vimirogant
RORγt, Ki: 3.5 nM
RORγt, IC50: 17 nM
    Selective Inhibitor
RORγt inverse agonist 13
ROR-γ, IC50: 63.8 nM
    Pan Inhibitor 99.22%