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Others

Related Products

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There are a number of inhibitors, agonists, and antagonists which we cannot make precise classification because the research area is still unknown.

Others Related Products (73734):

Cat. No. Product Name CAS No. Purity Chemical Structure
  • HY-108608
    o-3M3FBS 313981-55-4 99.79%
    o-3M3FBS is the negative control of m-3M3FBS. o-3M3FBS inhibits inward and outward currents via mechanisms independent of PLC acting in an antagonistic manner. In contrast, o-3M3FBS also causes an increase in [Ca2+]i in an agonistic manner.
    o-3M3FBS
  • HY-111082
    ISAM-140 932191-62-3 99.13%
    ISAM-140 (22b) is a potent and highly selective A2B adenosine receptor antagonist with a Ki of 3.49 nM.
    ISAM-140
  • HY-111083
    ML191 931695-79-3 99.81%
    ML-191 is an antagonist of GPR55. It inhibits GPR55 signaling induced by lysophosphatidylinositol (EC50=1.076 µM in U2OS cells overexpressing GPR55). ML-191 inhibits LPI-induced phosphorylation of ERK1/2 (IC50=328 nM) and receptor-dependent translocation of PKCβII when used at a concentration of 30 µM.
    ML191
  • HY-111616
    GSK1820795A 2650253-86-2 99.80%
    GSK1820795A, as a telmisartan analog, is a selective hGPR132a antagonist. GSK1820795A blocks activation of yeast cells expressing hGPR132a by N-acylamides. GSK1820795A is also a angiotensin II antagonists and partial PPARγ agonists (compound 38).
    GSK1820795A
  • HY-111934
    Cymarin 508-77-0
    Cymarin, a cardiac glycoside, potently inhibits the Palytoxin (PTX)-induced K+ release (IC50=0.42 μM). Cymarin reveals an antitumor activity against breast cancer and pancreatic cancer. Cymarin exhibits antifeedant and growth inhibitory effects as crop protectant.
    Cymarin
  • HY-112648
    Stafib-2 2097938-74-2 99.97%
    Stafib-2 is a potent and selctive inhibitor of the transcription factor STAT5b, with an IC50 of 82 nM and 1.7 μM for STAT5b and STAT5a, respectively. Stafib-2 exhibits poor cell permeability.
    Stafib-2
  • HY-113101
    2-Hydroxyadipic acid 18294-85-4 99.38%
    2-Hydroxyadipic acid is a dicarboxylic acid and monomer for functional polymers.2-Hydroxyadipic acid bears structural similarity to adipic acid.2-Hydroxyadipic acid forms via oxidative C-C cleavage of 2-hydroxycyclohexanone as a sustainable monomer source.
    2-Hydroxyadipic acid
  • HY-113302
    19-Hydroxyandrost-4-ene-3,17-dione 510-64-5 99.11%
    19-Hydroxyandrost-4-ene-3,17-dione is a substrate for Corticotropin-lipotropin and Cytochrome P450 19A1.
    19-Hydroxyandrost-4-ene-3,17-dione
  • HY-114362
    DL-alpha-Tocopherol methoxypolyethylene glycol succinate 1309573-60-1 98.14%
    DL-alpha-Tocopherol methoxypolyethylene glycol succinate (TPGS-750-M) is an amphiphile, acts as a surfactant. DL-alpha-Tocopherol methoxypolyethylene glycol succinate has a positive effect on Suzuki-Miyaura cross coupling. DL-alpha-Tocopherol methoxypolyethylene glycol succinate increases the styrene titer. DL-alpha-Tocopherol methoxypolyethylene glycol succinate is used in the stability test of NPYM-modified drugs in biological fluids.
    DL-alpha-Tocopherol methoxypolyethylene glycol succinate
  • HY-118075
    Coenzyme Q2 606-06-4
    Coenzyme Q2 is a biochemical reagent that can be used as a biological material or organic compound for life science related research.
    Coenzyme Q2
  • HY-120177
    KT182 1402612-62-7 ≥99.0%
    KT182 is a potent and selective inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.24 nM in Neuro2A cells.
    KT182
  • HY-122410
    Dihydrolanosterol 79-62-9 99.72%
    Dihydrolanosterol is a subtrate of CYP51 and a cholesterol biosynthesis inhibitor..
    Dihydrolanosterol
  • HY-123749
    Tetramethylrhodamine-5-iodoacetamide 114458-99-0
    Tetramethylrhodamine-5-iodoacetamide (5-TMRIA) is a thiol-selective reactive dye that is used to non-specifically label proteins via the cysteine residues. Tetramethylrhodamine-5-iodoacetamide (5-TMRIA) can be used to covalently label DNA fragments.
    Tetramethylrhodamine-5-iodoacetamide
  • HY-126411
    Peonidin-3-O-galactoside chloride 28148-89-2
    Peonidin-3-O-galactoside chloride is an anthocyanin with antioxidant properties and blood-brain barrier permeability. Peonidin-3-O-galactoside chloride inhibits pancreatic lipase, with an IC50 value of 23.2 μg/mL against porcine pancreatic lipase. Peonidin-3-O-galactoside chloride mediates neuroprotection, regulates glucose metabolism, protects cells from high glucose-induced damage, promotes glucose uptake and increases ATP production. Peonidin-3-O-galactoside (chloride) can be used in the research of obesity and neurodegenerative diseases.
    Peonidin-3-O-galactoside chloride
  • HY-126558
    GA3-AM 1373154-68-7 99.62%
    GA3-AM is a cell permeable analog of the plant hormone gibberellic acid that acts as a chemical dimerizer or chemical inducer of dimerization.
    GA3-AM
  • HY-126994
    6′-Amino-D-luciferin 161055-47-6 98.45%
    6’-Amino-D-luciferin is a derivative of D-luciferin (HY-12591A) with an amino group replacing the 6-hydroxyl group. 6’-Amino-D-luciferin is a natural substrate of luciferase (Luc) and can be used for IVIS imaging in cell/animal experiments[1][2][3].
    6′-Amino-D-luciferin
  • HY-129126
    NC9 1352090-52-8 99.98%
    NC9 (Cbz-Lys(Acr)-PEG2-dansyl) is an irreversible transglutaminase (TG) inhibitor. NC9 inhibits osteoblast differentiation and mineralization. NC9 destabilizes microtubules. NC9 can be used for the research of osteoblast differentiation.
    NC9
  • HY-130189
    S-Phenylmercapturic acid 4775-80-8 99.38%
    S-Phenylmercapturic acid, a metabolite of benzene, can be used as a biomarker, identified by GC, HPLC (UV or fluorescence detection), GC-MS, LC-MS/MS or immunoassay.
    S-Phenylmercapturic acid
  • HY-130433
    NBD Sphingosine 1449370-25-5 ≥99.0%
    NBD Sphingosine (NBD-Sph), a fluorochrome, is a fluorescence-labeled sphingosine. NBD Sphingosine can be uesd for fluorescence assay for sphingosine kinases.
    NBD Sphingosine
  • HY-131021
    Janelia Fluor® 549, Azide 99.49%
    Janelia Fluor? 549, Azide (JF549, Azide) is a fluorescent dye with the absorption maximum (λab (max)) of 549 nm and emission maximum (λem (max)) of 571 nm. Janelia Fluor? products are licensed under U.S. Pat. Nos. 9,933,417, 10,018,624 and 10,161,932 and other patents from Howard Hughes Medical Institute. It contains an azide group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing alkyne groups. It can also undergo ring strain-promoted alkyne-azide cycloaddition (SPAAC) with molecules containing DBCO or BCN groups.
    Janelia Fluor® 549, Azide