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Results for "

2-amino-1-

" in MedChemExpress (MCE) Product Catalog:

By Targets:	Amino Acid Derivatives (2) Amyloid-β (1) Antibiotic (1) Apoptosis (1) Bacterial (1) Biochemical Assay Reagents (7) Ceramidase (1) Drug Derivative (3) Drug Intermediate (3) Endogenous Metabolite (1) Endothelin Receptor (1) Ephrin Receptor (1) GCGR (1) GnRH Receptor (1) Herbicide (1) Insulin Receptor (1) Isotope-Labeled Compounds (7) Melanocortin Receptor (1) MOFs (9) Nucleoside Antimetabolite/Analog (4) Parasite (1) PROTAC Linkers (1) PSMA (2) Radionuclide-Drug Conjugates (RDCs) (4) Reference Standards (6) Renin (1) Somatostatin Receptor (5)
By Research Areas:	Cancer (13) Cardiovascular Disease (1) Endocrinology (2) Infection (2) Metabolic Disease (5) Neurological Disease (8)
Oligonucleotides:	Nucleoside Analogs (3) Cytidine (2)

Inhibitors & Agonists

Biochemical Assay Reagents

Peptides

Natural
Products

Isotope-Labeled Compounds

Oligonucleotides

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-118716

PhIP 1 Publications Verification 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine	Others	Cancer
PhIP (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine) is the most abundant of generation of heterocyclic amines (HCA), resulted in the cooking of meat . DNA damaging and mutagenic activities. PhIP also has oestrogenic activity that could contribute to its tissue specific carcinogenicity .

HY-P4070

Insulin icodec	Insulin Receptor	Metabolic Disease
Insulin icodec is an Insulin (HY-P0035) analog that strongly but reversibly binds to albumin. Insulin icodec has long plasma half-life. Insulin icodec modulates insulin receptor activity, controls blood glucose levels, reduces HbA_1c levels, and binds reversibly to human serum albumin. Insulin icodec can be used for the research of type 2 diabetes mellitus .

HY-76274

*(1S,2R)-2-Amino-1,2-diphenylethanol*	Biochemical Assay Reagents	Others
(1S,2R)-2-Amino-1,2-diphenylethanol is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-59132

2-Amino-1-phenylethanol	Endogenous Metabolite Drug Intermediate	Infection
2-Amino-1-phenylethanol is a Norepinephrine (HY-13715) analog. 2-Amino-1-phenylethanol derivatives exhibit antimalarial activity against Plasmodium falciparum .

HY-P5362

NODAGA-LM3	Radionuclide-Drug Conjugates (RDCs) Somatostatin Receptor	Neurological Disease Cancer
NODAGA-LM3 is a ligand that can cross the blood-brain barrier and targets somatostatin receptor SSTR2 with high affinity (IC₅₀ = 1.3 nM). NODAGA-LM3 does not trigger the internalization of SSTR2 and can inhibit agonist-induced internalization processes. NODAGA-LM3 shows low uptake in normal tissues such as the liver and spleen, but high uptake in the lungs and blood pool. ⁶⁸Ga-labeled NODAGA-LM3 can serve as a PET imaging agent for well-differentiated neuroendocrine tumors, and is applied in studies related to small cell lung cancer and well-differentiated neuroendocrine tumors .

HY-P2336A

CCZ01048 TFA 3 Publications Verification	Melanocortin Receptor	Cancer
CCZ01048 TFA, a α-MSH analogue, exhibits high binding affinity to melanocortin 1 receptor (MC1R) with a K_i of 0.31 nM. CCZ01048 TFA shows rapid internalization into B16F10 melanoma cells and high in vivo stability. CCZ01048 TFA is a promising candidate for PET imaging of malignant melanoma .

HY-W688565

*(2S)-2-Amino-1-hydroxyoctadecan-3-one*	Ceramidase	Metabolic Disease
(2S)-2-Amino-1-hydroxyoctadecan-3-one is the product generated by the decarboxylative condensation of L-serine and palmitoyl-CoA catalyzed by serine palmitoyltransferase (SPT) .

HY-W007825

*(1R,2S)-2-Amino-1,2-diphenylethanol*	Biochemical Assay Reagents	Others
(1R,2S)-2-Amino-1,2-diphenylethanol is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-Y0168

L-(-)-Phenylalaninol (S)-3-Phenyl-2-amino-1-propanol; (S)-Phenylalaninol	Amino Acid Derivatives	Others
L-(-)-Phenylalaninol is an alanine derivative .

HY-Y0837

L-Alaninol (S)-2-amino-1-propanol; (S)-2-aminopropanol; (S)-Alaninol	Biochemical Assay Reagents	Others
L-Alaninol is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-P10341

ZP3022	GCGR	Metabolic Disease
ZP3022 is a dual agonist of glucagon-like peptide-1 (GLP-1) and gastrin that has the ability to sustainably improve glycemic control. Additionally, ZP3022 can effectively increase β-cell mass, promote β-cell proliferation, and enhance the function of pancreatic islets. ZP3022 can be used in anti-diabetic research .

HY-79548

(+)-1,2-Diphenylethylenediamine (+)-Stilbenediamine	Biochemical Assay Reagents	Others
((1R,2R)-2-Amino-1,2-diphenylethyl)amine is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-Y0837S

L-Alaninol-d3 (S)-2-amino-1-propanol-d₃; (S)-2-aminopropanol-d₃; (S)-Alaninol-d₃	Isotope-Labeled Compounds	Others
L-Alaninol-d₃ is the deuterium labeled L-Alaninol .

HY-116443

2-Amino-1-phenylbutane hydrochloride	Drug Derivative	Neurological Disease
2-Amino-1-phenylbutane hydrochloride is an Amphetamine characterized by having an ethyl group in the alpha position .

HY-23212A

2-Amino-1,3-bis(carboxylethoxy)propane hydrochloride	Amino Acid Derivatives	Cancer
2-Amino-1,3-bis(carboxylethoxy)propane hydrochloride is a non-protein amino acid, sulfamic acid.2-Amino-1,3-bis(carboxylethoxy)propane hydrochloride contains one amino group and two terminal carboxylic acids.2-Amino-1,3-bis(carboxylethoxy)propane hydrochloride has a variety of physiological functions, including maintaining the stability of cell membranes, regulating cholesterol metabolism, supporting the normal function of the nervous system, participating in collagen synthesis, and anti-oxidation .

HY-76089

*tert-Butyl 3-(1-amino-2-methylpropan-2-yl)-1H-indole-1-carboxylate* 3-(2-amino-1,1-dimethylethyl)-indole-1-carboxylic acid tert-butyl ester	Drug Intermediate	Others
tert-Butyl 3-(1-amino-2-methylpropan-2-yl)-1H-indole-1-carboxylate (3-(2-Amino-1,1-dimethylethyl)-indole-1-carboxylic acid tert-butyl ester) is a drug intermediate for synthesis of various active compounds.

HY-152877

Isocytidine	Nucleoside Antimetabolite/Analog	Others
2-Amino-1-β-D-ribofuranosyl-4(1H)-pyrimidinone is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc .

HY-W391574

2-Amino-1-(3-chlorophenyl)-1-propanone hydrochloride	Drug Derivative	Neurological Disease
2-Amino-1-(3-chlorophenyl)-1-propanone hydrochloride is a drug derivative.

HY-118716S

PhIP-d3 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine-d₃	Isotope-Labeled Compounds	Cancer
PhIP-d₃ (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine-d₃) is the deuterium labeled PhIP (HY-118716). PhIP (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine) is the most abundant of generation of heterocyclic amines (HCA), resulted in the cooking of meat . DNA damaging and mutagenic activities. PhIP also has oestrogenic activity that could contribute to its tissue specific carcinogenicity .

HY-23212

2-Amino-1,3-bis(carboxylethoxy)propane	PROTAC Linkers	Cancer
2-Amino-13-bis(carboxylethoxy)propane is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-W007357R

2-Aminopropane-1,3-diol (Standard) 2-amino-1,3-propanediol (Standard)	Reference Standards
2-Aminopropane-1,3-diol (Standard) is the analytical standard of 2-Aminopropane-1,3-diol. This product is intended for research and analytical applications.

HY-P11004

A3-APO	Bacterial Antibiotic	Infection
A3-APO is an antimicrobial peptide. A3-APO has a significant antimicrobial activity by a dual mode of action with both membrane disintegration and intracellular target inhibition. A3-APO can deactivate bacterial toxins and increase the expression of anti-inflammatory cytokines (such as IL-4 and IL-10), without antimicrobial resistance. A3-APO accelerates burn wounds healing in mice infection model of Acinetobacter baumannii and Staphylococcus aureus .

HY-P10472

Azaline B	GnRH Receptor	Endocrinology
Azaline B is an antagonist for gonadotropin-releasing hormone (GnRH) with IC₅₀ of 1.37 nM, Azaline B can be used in research of sex hormone-related pathological states, ovulation induction and male contraception .

HY-P4757

N1-Glutathionyl-spermidine disulfide	Parasite	Others
N1-Glutathionyl-spermidine disulfide is a substrate of trypanothione reductase .

HY-21376S

*tert-Butyl 4-amino-1H-pyrazole-1-carboxylate-d2*	Isotope-Labeled Compounds	Others
tert-Butyl 4-amino-1H-pyrazole-1-carboxylate-d₂ is the deuterium labeled tert-Butyl 4-amino-1H-pyrazole-1-carboxylate.

HY-P11243

EphA4 agonist compound 23	Ephrin Receptor	Neurological Disease
EphA4 agonist compound 23 is a novel EphA4 agonist peptide mimic. EphA4 agonist compound 23 exhibits high affinity, high selectivity, and significant receptor activation ability. EphA4 agonist compound 23 is commonly used in the study of neurodegenerative diseases .

HY-P2434

AP102	Somatostatin Receptor	Neurological Disease Metabolic Disease Cancer
AP102 is a dual SSTR2/SSTR5-specific somatostatin analog (SSA). AP102 is a disulfide-bridged octapeptide SSA containing synthetic iodinated amino acids. AP102 binds with subnanomolar affinity to SSTR2 and SSTR5 (IC₅₀: 0.63 and 0.65 nM, respectively). AP102 does not bind to SSTR1 or SSTR3. AP102 can be used for acromegaly and neuroendocrine tumors research .

HY-P5362A

NODAGA-LM3 TFA	Radionuclide-Drug Conjugates (RDCs) Somatostatin Receptor	Cancer
NODAGA-LM3 TFA is a ligand that can cross the blood-brain barrier and targets somatostatin receptor SSTR2 with high affinity (IC₅₀ = 1.3 nM). NODAGA-LM3 TFA does not trigger the internalization of SSTR2 and can inhibit agonist-induced internalization processes. NODAGA-LM3 TFA shows low uptake in normal tissues such as the liver and spleen, but high uptake in the lungs and blood pool. ⁶⁸Ga-labeled NODAGA-LM3 TFA can serve as a PET imaging agent for well-differentiated neuroendocrine tumors, and is applied in studies related to small cell lung cancer and well-differentiated neuroendocrine tumors .

HY-105168

TAK 044	Endothelin Receptor	Cardiovascular Disease
TAK 044 is an antagonist of Endothelin Receptor. TAK 044 strongly inhibits ET-induced deterioration in various animal models. TAK 044 can be used in study ET-related diseases such as acute myocardial infarction,acute renal failure, acute hepatic malfunction, and subarachnoid hemorrhage .

HY-59132R

2-Amino-1-phenylethanol (Standard)	Reference Standards Drug Intermediate	Others
2-Amino-1-phenylethanol (Standard) is the analytical standard of 2-Amino-1-phenylethanol. This product is intended for research and analytical applications. 2-Amino-1-phenylethanol is a pharmaceutical intermediate that can be used for the synthesis of antimalarial agents and β₂-adrenergic receptor agonists.

HY-W173408

2-Amino-1-(4-chlorophenyl)propan-1-one hydrochloride	Drug Derivative	Neurological Disease
2-Amino-1-(4-chlorophenyl)propan-1-one hydrochloride is a drug derivative.

HY-W742257

2-Amino-1-(p-tolyl)ethanol-d3 Benzenemethanol, a-(aminomethyl)-4-methyl-d3	Isotope-Labeled Compounds	Others
2-Amino-1-(p-tolyl)ethanol-d₃ (Benzenemethanol, a-(aminomethyl)-4-methyl-d₃) is the deuterium labeled 2-Amino-1-(p-tolyl)ethanol (HY-W259001).

HY-W002642

2-Amino-1-cyclopentene-1-carbonitrile 2-aminocyclopent-1-ene-1-carbonitrile	Biochemical Assay Reagents	Others
2-Amino-1-cyclopentene-1-carbonitrile (2-Aminocyclopent-1-ene-1-carbonitrile) is an important and universal synthetic intermediate in organic chemistry.

HY-152603

2-Amino-1-β-D-arabinofuranosyl-5-methyl-4(1H)-pyrimidinone	Nucleoside Antimetabolite/Analog	Others
2-Amino-1-β-D-arabinofuranosyl-5-methyl-4(1H)-pyrimidinone is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc .

HY-118716R

PhIP (Standard) 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (Standard)	Others Reference Standards	Cancer
PhIP (Standard) is the analytical standard of PhIP. This product is intended for research and analytical applications. PhIP (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine) is the most abundant of generation of heterocyclic amines (HCA), resulted in the cooking of meat . DNA damaging and mutagenic activities. PhIP also has oestrogenic activity that could contribute to its tissue specific carcinogenicity .

HY-121504A

2-Amino-1-(4-methylphenyl)-1-propanone hydrochloride	Biochemical Assay Reagents	Neurological Disease
4-Methylcathinone (Normephedrone) hydrochloride is a drug derivative with neurostimulatory activity .

HY-Z6843R

Noradrenalone impurity 1 hydrochloride (Standard)	Reference Standards
2-Amino-1-(3,4-dihydroxyphenyl)ethanone hydrochloride (Noradrenaline Impurity) (Standard) is the analytical standard of 2-Amino-1-(3,4-dihydroxyphenyl)ethanone hydrochloride (Noradrenaline Impurity). This product is intended for research and analytical applications.

HY-P2075

EMD 55068	Renin	Endocrinology
EMD 55068 is a renin antagonist. EMD 55068 inhibits the uptake of taurocholate .

HY-152878

Arabinosylisocytosine NSC 529488	Nucleoside Antimetabolite/Analog	Others
2-Amino-1-β-D-arabinofuranosyl-4(1H)-pyrimidinone is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc .

HY-P10876

mcK6A1	Amyloid-β	Neurological Disease
mcK6A1 is an inhibitor for the aggregation of amyloid-β (Aβ), that selectively binds to the 16KLVFFA21 segment of Aβ42, forms an extended β-folded structure, and inhibits the formation of Aβ42 oligomers. mcK6A1 can be used in research of Alzheimer's disease and other amyloid-related diseases .

HY-W770415

D,L-N,N-Didesmethyl Venlafaxine-d11	Isotope-Labeled Compounds	Others
D,L-N,N-Didesmethyl Venlafaxine-d₁₁ is the deuterium labeled 1-(2-Amino-1-(4-methoxyphenyl)ethyl)cyclohexan-1-ol (HY-W317961).

HY-N14253

*cis-2-Amino-1-hydroxycyclobutane-1-acetic acid*	Herbicide	Others
cis-2-Amino-1-hydroxycyclobutane-1-acetic acid is a herbicidal antimetabolite that can cause L-cysteineor L-methionine-reversible chlorosis in Arabidopsis thaliana .

HY-W308027

*(2-Amino-1-hydroxyethyl)phosphonate* 1-Hydroxy-2-aminoethylphosphonic acid	Nucleoside Antimetabolite/Analog	Metabolic Disease
(2-Amino-1-hydroxyethyl)phosphonate (1-Hydroxy-2-aminoethylphosphonic acid) is a nucleoside metabolite.

HY-W703677

2-Amino-1-(p-tolyl)ethan-1-one hydrochloride-d3	Isotope-Labeled Compounds	Others
2-Amino-1-(p-tolyl)ethan-1-one hydrochloride-d₃ is the deuterium labeled 2-Amino-1-(p-tolyl)ethan-1-one hydrochloride (HY-W086589).

HY-W097771R

*1-(2-Amino-1-(4-methoxyphenyl)ethyl)cyclohexan-1-ol hydrochloride (Standard)*	Reference Standards
1-[2-Amino-1-(4-methoxyphenyl)ethyl]cyclohexanol Hydrochloride (Standard) is the analytical standard of 1-[2-Amino-1-(4-methoxyphenyl)ethyl]cyclohexanol Hydrochloride. This product is intended for research and analytical applications.

HY-W583350

*Chloro(triphenylphosphine) [2-(2'-amino-1,1'-biphenyl)]palladium(II)*	Apoptosis	Cancer
Chloro(triphenylphosphine)[2-(2'-amino-1,1'-biphenyl)]palladium(II) (Compound 4C) is a metal palladium (II) complex. Chloro(triphenylphosphine)[2-(2'-amino-1,1'-biphenyl)]palladium(II) exhibits potent anti-proliferative activity against cells such as MDA-MB-231 and HCT116, significantly inducing apoptosis. Chloro(triphenylphosphine)[2-(2'-amino-1,1'-biphenyl)]palladium(II) does not directly damage DNA or cause significant cell cycle arrest. Chloro(triphenylphosphine)[2-(2'-amino-1,1'-biphenyl)]palladium(II) can be used in studies on Cisplatin (HY-17394) resistance .

HY-W112579

2'-Amino-[1,1':3',1''-terphenyl]-4,4''-dicarboxylic acid	MOFs	Others
2'-Amino-[1,1':3',1''-terphenyl]-4,4''-dicarboxylic acid is a metal-organic framework (MOF).

HY-W075220

2'-Amino-[1,1':4',1''-terphenyl]-4,4''-dicarboxylic acid	MOFs	Others
2'-Amino-[1,1':4',1''-terphenyl]-4,4''-dicarboxylic acid is a metal-organic framework (MOF).

HY-W190904

2-Amino-1,3-bis(tert-butyldimethylsilanoxy)propane	Biochemical Assay Reagents	Others
2-Amino-1,3-bis(tert-butyldimethylsilanoxy)propane has a TBDMS, acid labile protecting group. TBDMS is used for the protection of alcohol groups. The primary amine is able to react with carboxylic acids, active NHS esters and other carbonyl compounds.

HY-W112947

2'-Amino-[1,1':3',1''-terphenyl]-4,4'',5'-tricarboxylicacid	MOFs	Others
2'-Amino-[1,1':3',1''-terphenyl]-4,4'',5'-tricarboxylicacid is a metal-organic framework (MOF).

Cat. No.	Product Name	Target	Research Area

HY-P4070

Insulin icodec	Insulin Receptor	Metabolic Disease
Insulin icodec is an Insulin (HY-P0035) analog that strongly but reversibly binds to albumin. Insulin icodec has long plasma half-life. Insulin icodec modulates insulin receptor activity, controls blood glucose levels, reduces HbA_1c levels, and binds reversibly to human serum albumin. Insulin icodec can be used for the research of type 2 diabetes mellitus .

HY-105055

Didemnin B	Peptides	Cancer
Didemnin B is a depsipeptide extracted from the marine tunicate Trididemnin cyanophorum. Didemnin B can be used for the research of cancer .

HY-P5362

NODAGA-LM3	Radionuclide-Drug Conjugates (RDCs) Somatostatin Receptor	Neurological Disease Cancer
NODAGA-LM3 is a ligand that can cross the blood-brain barrier and targets somatostatin receptor SSTR2 with high affinity (IC₅₀ = 1.3 nM). NODAGA-LM3 does not trigger the internalization of SSTR2 and can inhibit agonist-induced internalization processes. NODAGA-LM3 shows low uptake in normal tissues such as the liver and spleen, but high uptake in the lungs and blood pool. ⁶⁸Ga-labeled NODAGA-LM3 can serve as a PET imaging agent for well-differentiated neuroendocrine tumors, and is applied in studies related to small cell lung cancer and well-differentiated neuroendocrine tumors .

HY-P2336A

CCZ01048 TFA 3 Publications Verification	Melanocortin Receptor	Cancer
CCZ01048 TFA, a α-MSH analogue, exhibits high binding affinity to melanocortin 1 receptor (MC1R) with a K_i of 0.31 nM. CCZ01048 TFA shows rapid internalization into B16F10 melanoma cells and high in vivo stability. CCZ01048 TFA is a promising candidate for PET imaging of malignant melanoma .

HY-Y0168

L-(-)-Phenylalaninol (S)-3-Phenyl-2-amino-1-propanol; (S)-Phenylalaninol	Amino Acid Derivatives	Others
L-(-)-Phenylalaninol is an alanine derivative .

HY-P10341

ZP3022	GCGR	Metabolic Disease
ZP3022 is a dual agonist of glucagon-like peptide-1 (GLP-1) and gastrin that has the ability to sustainably improve glycemic control. Additionally, ZP3022 can effectively increase β-cell mass, promote β-cell proliferation, and enhance the function of pancreatic islets. ZP3022 can be used in anti-diabetic research .

HY-P11004

A3-APO	Bacterial Antibiotic	Infection
A3-APO is an antimicrobial peptide. A3-APO has a significant antimicrobial activity by a dual mode of action with both membrane disintegration and intracellular target inhibition. A3-APO can deactivate bacterial toxins and increase the expression of anti-inflammatory cytokines (such as IL-4 and IL-10), without antimicrobial resistance. A3-APO accelerates burn wounds healing in mice infection model of Acinetobacter baumannii and Staphylococcus aureus .

HY-P10472

Azaline B	GnRH Receptor	Endocrinology
Azaline B is an antagonist for gonadotropin-releasing hormone (GnRH) with IC₅₀ of 1.37 nM, Azaline B can be used in research of sex hormone-related pathological states, ovulation induction and male contraception .

HY-P4757

N1-Glutathionyl-spermidine disulfide	Parasite	Others
N1-Glutathionyl-spermidine disulfide is a substrate of trypanothione reductase .

HY-P11243

EphA4 agonist compound 23	Ephrin Receptor	Neurological Disease
EphA4 agonist compound 23 is a novel EphA4 agonist peptide mimic. EphA4 agonist compound 23 exhibits high affinity, high selectivity, and significant receptor activation ability. EphA4 agonist compound 23 is commonly used in the study of neurodegenerative diseases .

HY-P2434

AP102	Somatostatin Receptor	Neurological Disease Metabolic Disease Cancer
AP102 is a dual SSTR2/SSTR5-specific somatostatin analog (SSA). AP102 is a disulfide-bridged octapeptide SSA containing synthetic iodinated amino acids. AP102 binds with subnanomolar affinity to SSTR2 and SSTR5 (IC₅₀: 0.63 and 0.65 nM, respectively). AP102 does not bind to SSTR1 or SSTR3. AP102 can be used for acromegaly and neuroendocrine tumors research .

HY-P5362A

NODAGA-LM3 TFA	Radionuclide-Drug Conjugates (RDCs) Somatostatin Receptor	Cancer
NODAGA-LM3 TFA is a ligand that can cross the blood-brain barrier and targets somatostatin receptor SSTR2 with high affinity (IC₅₀ = 1.3 nM). NODAGA-LM3 TFA does not trigger the internalization of SSTR2 and can inhibit agonist-induced internalization processes. NODAGA-LM3 TFA shows low uptake in normal tissues such as the liver and spleen, but high uptake in the lungs and blood pool. ⁶⁸Ga-labeled NODAGA-LM3 TFA can serve as a PET imaging agent for well-differentiated neuroendocrine tumors, and is applied in studies related to small cell lung cancer and well-differentiated neuroendocrine tumors .

HY-105168

TAK 044	Endothelin Receptor	Cardiovascular Disease
TAK 044 is an antagonist of Endothelin Receptor. TAK 044 strongly inhibits ET-induced deterioration in various animal models. TAK 044 can be used in study ET-related diseases such as acute myocardial infarction,acute renal failure, acute hepatic malfunction, and subarachnoid hemorrhage .

HY-P2075

EMD 55068	Renin	Endocrinology
EMD 55068 is a renin antagonist. EMD 55068 inhibits the uptake of taurocholate .

HY-P10876

mcK6A1	Amyloid-β	Neurological Disease
mcK6A1 is an inhibitor for the aggregation of amyloid-β (Aβ), that selectively binds to the 16KLVFFA21 segment of Aβ42, forms an extended β-folded structure, and inhibits the formation of Aβ42 oligomers. mcK6A1 can be used in research of Alzheimer's disease and other amyloid-related diseases .

HY-P11488

JR11-PEG3-DOTA-PSMA-03	Radionuclide-Drug Conjugates (RDCs) Somatostatin Receptor PSMA	Cancer
JR11-PEG3-DOTA-PSMA-03 (Compound 2) is an RDC-related compound containing the chelating agent DOTA (HY-W053583), the JR11 peptide (SSTR2 antagonist), and the PSMA ligand. JR11-PEG3-DOTA-PSMA-03 shows SSTR2-binding affinities and PSMA-binding affinities, with IC₅₀ s of 94.0 nM, 81.8 nM, respectively. JR11-PEG3-DOTA-PSMA-03 can be radiolabeled with [ ⁶⁸Ga]. [ ⁶⁸Ga] radiolabeled JR11-PEG3-DOTA-PSMA-03 can be used in diagnostic studies of neuroendocrine differentiated prostate cancer .

HY-P11485

JR11-PEG3-HBED-CC-PSMA-03	Radionuclide-Drug Conjugates (RDCs) Somatostatin Receptor PSMA	Cancer
JR11-PEG3-HBED-CC-PSMA-03 (Compound 1) is an RDC-related compound containing the chelating agent HBED-CC, the JR11 peptide (SSTR2 antagonist), and the PSMA ligand. JR11-PEG3-HBED-CC-PSMA-03 shows SSTR2-binding affinities and PSMA-binding affinities, with IC₅₀ s of 59.2 nM, 57.0 nM, respectively. JR11-PEG3-HBED-CC-PSMA-03 can be radiolabeled with [ ⁶⁸Ga]. [ ⁶⁸Ga] radiolabeled JR11-PEG3-HBED-CC-PSMA-03 can be used in diagnostic studies of neuroendocrine differentiated prostate cancer .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-118716

PhIP 1 Publications Verification 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine	Human Gut Microbiota Metabolites Endogenous metabolite Source Classification	Others
PhIP (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine) is the most abundant of generation of heterocyclic amines (HCA), resulted in the cooking of meat . DNA damaging and mutagenic activities. PhIP also has oestrogenic activity that could contribute to its tissue specific carcinogenicity .

HY-105055

Didemnin B	Natural Products Animals Classification of Application Fields Marine natural products Other marine organisms Disease Research Fields Source Classification Cancer	Others
Didemnin B is a depsipeptide extracted from the marine tunicate Trididemnin cyanophorum. Didemnin B can be used for the research of cancer .

HY-59132

2-Amino-1-phenylethanol	Natural Products Classification of Application Fields Other Diseases Endogenous metabolite Disease Research Fields Source Classification	Endogenous Metabolite Drug Intermediate
2-Amino-1-phenylethanol is a Norepinephrine (HY-13715) analog. 2-Amino-1-phenylethanol derivatives exhibit antimalarial activity against Plasmodium falciparum .

HY-Y0837

L-Alaninol (S)-2-amino-1-propanol; (S)-2-aminopropanol; (S)-Alaninol	Microorganisms Source Classification	Biochemical Assay Reagents
L-Alaninol is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-59132R

2-Amino-1-phenylethanol (Standard)	Structural Classification Natural Products Endogenous metabolite Source Classification	Reference Standards Drug Intermediate
2-Amino-1-phenylethanol (Standard) is the analytical standard of 2-Amino-1-phenylethanol. This product is intended for research and analytical applications. 2-Amino-1-phenylethanol is a pharmaceutical intermediate that can be used for the synthesis of antimalarial agents and β₂-adrenergic receptor agonists.

HY-N14253

*cis-2-Amino-1-hydroxycyclobutane-1-acetic acid*	Natural Products Microorganisms Source Classification	Herbicide
cis-2-Amino-1-hydroxycyclobutane-1-acetic acid is a herbicidal antimetabolite that can cause L-cysteineor L-methionine-reversible chlorosis in Arabidopsis thaliana .

HY-W308027

*(2-Amino-1-hydroxyethyl)phosphonate* 1-Hydroxy-2-aminoethylphosphonic acid	Structural Classification Natural Products Amino acids Endogenous metabolite Source Classification	Nucleoside Antimetabolite/Analog
(2-Amino-1-hydroxyethyl)phosphonate (1-Hydroxy-2-aminoethylphosphonic acid) is a nucleoside metabolite.

Cat. No.	Product Name	Chemical Structure

HY-Y0837S

L-Alaninol-d3
L-Alaninol-d₃ is the deuterium labeled L-Alaninol .

HY-118716S

PhIP-d3

PhIP-d₃ (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine-d₃) is the deuterium labeled PhIP (HY-118716). PhIP (2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine) is the most abundant of generation of heterocyclic amines (HCA), resulted in the cooking of meat . DNA damaging and mutagenic activities. PhIP also has oestrogenic activity that could contribute to its tissue specific carcinogenicity .

HY-21376S

*tert-Butyl 4-amino-1H-pyrazole-1-carboxylate-d2*
tert-Butyl 4-amino-1H-pyrazole-1-carboxylate-d₂ is the deuterium labeled tert-Butyl 4-amino-1H-pyrazole-1-carboxylate.

HY-W742257

2-Amino-1-(p-tolyl)ethanol-d3
2-Amino-1-(p-tolyl)ethanol-d₃ (Benzenemethanol, a-(aminomethyl)-4-methyl-d₃) is the deuterium labeled 2-Amino-1-(p-tolyl)ethanol (HY-W259001).

HY-W770415

D,L-N,N-Didesmethyl Venlafaxine-d11
D,L-N,N-Didesmethyl Venlafaxine-d₁₁ is the deuterium labeled 1-(2-Amino-1-(4-methoxyphenyl)ethyl)cyclohexan-1-ol (HY-W317961).

HY-W703677

2-Amino-1-(p-tolyl)ethan-1-one hydrochloride-d3
2-Amino-1-(p-tolyl)ethan-1-one hydrochloride-d₃ is the deuterium labeled 2-Amino-1-(p-tolyl)ethan-1-one hydrochloride (HY-W086589).

HY-W013029S

(S)-2-Aminobutan-1-ol-d6
(S)-2-Aminobutan-1-ol-d₆ (S-(+)-2-Amino-1-butanol-d₆) is the deuterium labeled (S)-2-Aminobutan-1-ol.

Cat. No.	Product Name		Classification

HY-152877

Isocytidine		Nucleoside Analogs Cytidine
2-Amino-1-β-D-ribofuranosyl-4(1H)-pyrimidinone is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc .

HY-152603

2-Amino-1-β-D-arabinofuranosyl-5-methyl-4(1H)-pyrimidinone		Nucleoside Analogs
2-Amino-1-β-D-arabinofuranosyl-5-methyl-4(1H)-pyrimidinone is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc .

HY-152878

Arabinosylisocytosine NSC 529488		Nucleoside Analogs Cytidine
2-Amino-1-β-D-arabinofuranosyl-4(1H)-pyrimidinone is a purine nucleoside analogue. Purine nucleoside analogs have broad antitumor activity targeting indolent lymphoid malignancies. Anticancer mechanisms in this process rely on inhibition of DNA synthesis, induction of apoptosis, etc .

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