JR11-PEG3-HBED-CC-PSMA-03
JR11-PEG3-HBED-CC-PSMA-03 (Compound 1) is an RDC-related compound containing the chelating agent HBED-CC, the JR11 peptide (SSTR2 antagonist), and the PSMA ligand. JR11-PEG3-HBED-CC-PSMA-03 shows SSTR2-binding affinities and PSMA-binding affinities, with IC50 s of 59.2 nM, 57.0 nM, respectively. JR11-PEG3-HBED-CC-PSMA-03 can be radiolabeled with [68Ga]. [68Ga] radiolabeled JR11-PEG3-HBED-CC-PSMA-03 can be used in diagnostic studies of neuroendocrine differentiated prostate cancer.
For research use only. We do not sell to patients.
- Formula: C127H163ClN24O36S2
- Molecular Weight:2701.38
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Radionuclide-Drug Conjugates (RDCs) Isoforms
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Biological Activity
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SSTR2 |
Chemical Information
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Molecular Weight 2701.38
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Formula C127H163ClN24O36S2
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Sequence
{Phe(p-Cl)}-cyclo({d-Cys}-Phe-{d-4-amino-Phe(carbamoyl)}-Lys-Thr-Cys){d-Tyr}-NH2-PEG3-HBED-CC-PSMA-03
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Sequence Shortening
{Phe(p-Cl)}-cyclo({d-Cys}-F-{d-4-amino-Phe(carbamoyl)}-KTC){d-Tyr}-NH2-PEG3-HBED-CC-PSMA-03
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
JR11-PEG3-HBED-CC-PSMA-03 Related Classifications
HY-P11485 Related Classifications
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