1. Anti-infection
    Metabolic Enzyme/Protease
    Membrane Transporter/Ion Channel
  2. HIV
    HIV Protease
    SARS-CoV
    Cytochrome P450
    P-glycoprotein
    Endogenous Metabolite
  3. Atazanavir

Atazanavir  (Synonyms: BMS-232632)

Cat. No.: HY-17367
Handling Instructions

Atazanavir (BMS-232632), a highly selective HIV-1 protease inhibitor, is the first protease inhibitor approved for once-daily administration. Atazanavir (BMS-232632) is a substrate and inhibitor of CYP3A4, and an inhibitor and inducer of P-glycoprotein (P-gp). Atazanavir is also a SARS-CoV 3CLpro inhibitor with an IC50 of 3.49 μM.

For research use only. We do not sell to patients.

Atazanavir Chemical Structure

Atazanavir Chemical Structure

CAS No. : 198904-31-3

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Description

Atazanavir (BMS-232632), a highly selective HIV-1 protease inhibitor, is the first protease inhibitor approved for once-daily administration[1]. Atazanavir (BMS-232632) is a substrate and inhibitor of CYP3A4, and an inhibitor and inducer of P-glycoprotein (P-gp)[2]. Atazanavir is also a SARS-CoV 3CLpro inhibitor with an IC50 of 3.49 μM[3].

IC50 & Target

CYP3

 

HIV-1

 

Clinical Trial
Molecular Weight

704.86

Formula

C38H52N6O7

CAS No.
SMILES

O=C(OC)N[[email protected]@H](C(C)(C)C)C(NN(CC1=CC=C(C2=NC=CC=C2)C=C1)C[[email protected]](O)[[email protected]](CC3=CC=CC=C3)NC([[email protected]](C(C)(C)C)NC(OC)=O)=O)=O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Atazanavir
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