36 Results for "

Deacetyl

" in MedChemExpress (MCE) Product Catalog:
Products (36)

36 Results for "Deacetyl" in MCE Product Catalog:

4
4 Cited Publications
Cat. No.: HY-P2161B
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM) with improved metabolic stability. TAK-683 acetate is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively . TAK-683 acetate depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer .
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Cat. No.: HY-G0018
CAS No.: 53016-31-2
Synonyms: 17-Deacetyl norgestimate; 17-Deacylnorgestimate
Target:  

Drug Metabolite

Research Areas:  

Endocrinology

Norgestimate metabolite Norelgestromin (17-Deacetyl norgestimate) is a metabolite of Norgestimate (HY-W013172). Norgestimate metabolite Norelgestromin is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
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Cat. No.: HY-20584
CAS No.: 90332-63-1
Synonyms: 10-Deacetyl-7-xylosyltaxol; 10-Deacetylpaclitaxel 7-Xyloside; 10-Deacetyltaxol 7-Xyloside
10-Deacetyl-7-xylosyl paclitaxel is a Paclitaxel (a microtubule stabilizing agent; enhances tubulin polymerization) derivative with improved pharmacological features.
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Cat. No.: HY-14959
CAS No.: 159811-51-5
Purity:  ≥98.0%
Synonyms: CDB-3236; Deacetyl CDB-2914
Target:  

Progesterone Receptor

Research Areas:  

Endocrinology Cancer

Ulipristal (CDB 3236) is a selective progesterone receptor modulator (SPRM). Ulipristal binds to the progesteron receptor, thereby inhibiting PR-mediated gene expression, and interfering with progesterone activity in the reproductive system .
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Cat. No.: HY-77572
CAS No.: 78454-17-8
Synonyms: 7-epi-10-Deacetyltaxol; 10-Deacetyl-7-epipaclitaxel
7-Epi 10-desacetyl paclitaxel (7-epi-10-deacetyltaxol), a taxol derivative, exhibits cytotoxicity against HeLa cells with an IC50 of 85 μM .
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Cat. No.: HY-P5544
CAS No.: 60230-21-9
Synonyms: N-Acetylmuramyl-L-Ala-γ-D-Glu-meso-diaminopimelic acid
Research Areas:  

Others

M-TriDAP (N-Acetylmuramyl-L-Ala-γ-D-Glu-meso-diaminopimelic acid) is a NOD1/2 agoist and biological active peptide .
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Cat. No.: HY-N3501
CAS No.: 100665-44-9
Deacetyl Ganoderic Acid F is a 7-anostane triterpenoid from Ganoderma lucidum.
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Cat. No.: HY-P2161
CAS No.: 872719-49-8
Target:  

Kisspeptin Receptor

Research Areas:  

Cancer

TAK-683 is a potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM) with improved metabolic stability. TAK-683 is a nonapeptide metastin analog, exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM and 1.6 nM for human and rat, respectively . TAK-683 depletes GnRH in the hypothalamus and reduces plasma FSH, LH, and testosterone levels in vivo, it has the potential for the study of hormone-dependent prostate cancer .
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Cat. No.: HY-Z8644
CAS No.: 7411-12-3
Synonyms: N-Formyl-N-Deacetylcolchicine
Research Areas:  

Cancer

N-Deacetyl-N-formylcolchicine (N-Formyl-N-deacetylcolchicine, Compound 11) is a selective inhibitor targeting the colchicine-binding site of tubulin. N-Deacetyl-N-formylcolchicine shows antiproliferative activity against various cancer cell lines with IC50 values of 32.61-100.28 nM. N-Deacetyl-N-formylcolchicine inhibits microtubule polymerization to block cell division, induces cancer cell apoptosis and suppresses migration. N-Deacetyl-N-formylcolchicine is promising for research of cancers such as lung cancer and various solid tumors .
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Cat. No.: HY-Z8147
CAS No.: 4701-54-6
Synonyms: 16-Deacetylfusidic acid γ-lactone
Target:  

Bacterial

Research Areas:  

Infection

16-O-Deacetyl fusidic acid lactone (16-Deacetylfusidic acid γ-lactone) (FA-9) is a Fusidic acid (HY-B1350) (FA) lactone derivative with antibacterial effects. 16-O-Deacetyl fusidic acid lactone is effective against Gram-positive bacteria, but has no inhibitory effect on Gram-negative bacteria .
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Cat. No.: HY-77572R
CAS No.: 78454-17-8
Synonyms: 7-epi-10-Deacetyltaxol (Standard); 10-Deacetyl-7-epipaclitaxel (Standard)
7-Epi 10-desacetyl paclitaxel (Standard) is the analytical standard of 7-Epi 10-desacetyl paclitaxel. This product is intended for research and analytical applications. 7-Epi 10-desacetyl paclitaxel (7-epi-10-deacetyltaxol), a taxol derivative, exhibits cytotoxicity against HeLa cells with an IC50 of 85 μM .
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Cat. No.: HY-G0018S
CAS No.: 1263184-13-9
Synonyms: 17-Deacetyl norgestimate-d6; 17-Deacylnorgestimate-d6
Norgestimate metabolite norelgestromin-d6 is the deuterium labeled Norgestimate metabolite norelgestromin. Norelgestromin is a metabolite of Norgestimate, which is a progestin or synthetic progestogen. Norgestimate metabolite norelgestromin-d6 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
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Cat. No.: HY-P2115
CAS No.: 127932-90-5
Target:  

GnRH Receptor

Research Areas:  

Cancer

Ramorelix is a luteinizing-hormone-releasing hormone (LHRH) antagonist. Ramorelix can inhibit tumor progression in vivo. Ramorelix can be studied in anti-cancer research .
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Cat. No.: HY-W778562
CAS No.: 92950-42-0
10-Deacetyl-13-oxobaccatin III is an taxane that can be isolated from Taxus sumatrana. 10-Deacetyl-13-oxobaccatin III (30 μg/mL) shows cytotoxicity against A498, NCI-H226, A549, PC-3 cells, with inhibition a rate of 29.7%, 49.2%, 43.9%, 65.3% .
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Cat. No.: HY-W778546
CAS No.: 71629-92-0
7-epi-10-Deacetyl baccatin III can be isolated from the degradation impurities in Docetaxel (HY-B0011) .
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Cat. No.: HY-N9222
CAS No.: 172486-22-5
9-Deacetyl-9-benzoyl-10-debenzoyltaxchinin A is a Diterpenoids product that can be isolated from the stem-barks of Taxus baccata L. cv. stricta. .
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Cat. No.: HY-N1640
CAS No.: 1189801-51-1
1-O-Deacetyl-2α-hydroxykhayanolide E is a natural product that can be isolated from Swietenia mahagoni. 1-O-Deacetyl-2α-hydroxykhayanolide E is widely distributed in the leaves and branches of Swietenia mahagoni .
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Cat. No.: HY-W778547
CAS No.: 151636-94-1
Synonyms: 10-Dehydrobaccatin V
7-epi-10-Oxo-10-deacetyl baccatin III (10-Dehydrobaccatin V) can be isolated from the degradation impurities in Docetaxel (HY-B0011) .
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Cat. No.: HY-N9033
CAS No.: 227011-48-5
9-Deacetyl-9-benzoyl-10-debenzoyl-4β,20-epoxytaxchinin A is a Diterpenoids product that can be isolated from the stem-barks of Taxus baccata L. cv. stricta. .
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Cat. No.: HY-125374A
CAS No.: 192573-38-9
Synonyms: XRP9881 dihydrate
Target:  

Microtubule/Tubulin

Research Areas:  

Cancer

Larotaxel (dihydrate) (XRP9881 (dihydrate)), a new taxane compound prepared by partial synthesis from 10-deacetyl baccatin III, is active against tumors .
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