2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. TRP Channel
  4. Capsiate

Capsiate, as a capsaicin analogue extracted from a non-pungent cultivar of CH-19 sweet red pepper, is an orally active agonist of TRPV1.

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Capsiate

Capsiate 構造式

CAS 番号 : 205687-01-0

容量 価格（税別） 在庫状況 数量
5 mg $230 在庫あり
10 mg $350 在庫あり
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Based on 4 publication(s) in Google Scholar

Capsiate 関連抗体

Top Publications Citing Use of Products

TRP Channel アイソフォーム固有の製品をすべて表示:

すべてのアイソフォームを表示
TRPA1 TRPC3 TRPC4 TRPC5 TRPC6 TRPC7 TRPM8 TRPM2 TRPM3 TRPM4 TRPM7 TRPML1 TRPML2 TRPML3 TRPV1 TRPV2 TRPV3 TRPV4 TRPV6

  • 生物活性

  • 純度とドキュメンテーション

  • 参考文献

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製品説明

Capsiate, as a capsaicin analogue extracted from a non-pungent cultivar of CH-19 sweet red pepper, is an orally active agonist of TRPV1[1].

IC50 & Target[1]

TRPV1

 

体外実験

Capsiate evokes current responses in HEK293 cells expressing TRPV1[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Capsiate 関連抗体
体内実験

Capsiate does not exhibit irritancy-related effects on the oral cavity or eye[1].
Capsiate (0.03~0.54 mM; s.c.) induces nociceptive responses in mice[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male ddY-strain mice (20–24 g) [1]
Dosage: 0.5 or 5 mM
Administration: P.o.
Result: Did not cause pungency-related behaviors.
臨床実験
分子量

306.40

分子式

C18H26O4
CAS 番号
Appearance

Liquid (Density: 1.053 g/cm3)

Color

Colorless to light yellow

SMILES

CC(C)/C=C/CCCCC(OCC1=CC=C(O)C(OC)=C1)=O
Structure Classification
Initial Source
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
溶剤 & 溶解度
体外: 

DMSO : 100 mg/mL (326.37 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.2637 mL 16.3185 mL 32.6371 mL
5 mM 0.6527 mL 3.2637 mL 6.5274 mL
10 mM 0.3264 mL 1.6319 mL 3.2637 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

一般には略語で表示されます：C1V1 = C2V2

濃度 （開始）

C1

×
体積 （開始）

V1

=
濃度 （終了）

C2

×
体積 （終了）

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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mg/kg

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(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
純度とドキュメンテーション

純度: 99.85%

COA (242 KB) HNMR (242 KB) LCMS (89 KB)

取扱説明書 (2659 KB)
参考文献

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 3.2637 mL 16.3185 mL 32.6371 mL 81.5927 mL
5 mM 0.6527 mL 3.2637 mL 6.5274 mL 16.3185 mL
10 mM 0.3264 mL 1.6319 mL 3.2637 mL 8.1593 mL
15 mM 0.2176 mL 1.0879 mL 2.1758 mL 5.4395 mL
20 mM 0.1632 mL 0.8159 mL 1.6319 mL 4.0796 mL
25 mM 0.1305 mL 0.6527 mL 1.3055 mL 3.2637 mL
30 mM 0.1088 mL 0.5440 mL 1.0879 mL 2.7198 mL
40 mM 0.0816 mL 0.4080 mL 0.8159 mL 2.0398 mL
50 mM 0.0653 mL 0.3264 mL 0.6527 mL 1.6319 mL
60 mM 0.0544 mL 0.2720 mL 0.5440 mL 1.3599 mL
80 mM 0.0408 mL 0.2040 mL 0.4080 mL 1.0199 mL
100 mM 0.0326 mL 0.1632 mL 0.3264 mL 0.8159 mL
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Capsiate Related Classifications

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

質量   濃度   体積   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

一般には略語で表示されます：C1V1 = C2V2

濃度 （開始） × 体積 （開始） = 濃度 （終了） × 体積 （終了）
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Capsiate205687-01-0TRP ChannelTransient receptor potential channelscapsaicinanaloguenon-pungentcultivarCH-19sweetredpepperInhibitorinhibitorinhibit

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製品名:
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製品番号:
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