1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
    Neuronal Signaling
  3. TRP Channel
  4. TRP Channel Inhibitors

TRP Channel Inhibitors

TRPM

TRPV

TRPA

TRPML

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

TRP Channel Inhibitors, Agonists, Antagonists & Activators
Product Name TRPM TRPV TRPA TRPML Purity
GSK1016790A  
TRPV4
    99.65%
SB-366791  
hTRPV1, IC50: 5.7 nM
    98.72%
(1R,2R)-ML-SI3      
TRPML1, IC50: 1.6 μM
TRPML2, IC50: 2.3 μM
TRPML3, IC50: 12.5 μM
98.15%
Dihydrocapsaicin  
TRPV1
    98.82%
RQ-00203078  
TRPV4, IC50: 10 μM
    99.84%
LE135  
TRPV1, EC50: 2.5 μM
TRPA1, EC50: 20 μM
  99.03%
ML-SI3      
TRPML1, IC50: 4.7 μM
99.81%
JNJ-17203212  
TRPV1
    99.94%
AS1269574    
TRPA1
  98.76%
MDR-652  
hTRPV1, Ki: 11.4 nM
rTRPV1, Ki: 23.8 nM
hTRPV1, EC50: 5.05 nM
rTRPV1, EC50: 93 nM
    98.17%
AP-18    
TRPA1, IC50: ~3 μM
  99.80%
Vanilloid receptor antagonist 1  
TRPV1
    98.07%
Chembridge-5861528    
TRPA1, IC50: 14.3 μM (allyl isothiocyanate-evoked TRPA1 response)
TRPA1, IC50: 18.7 μM (4-HNE-evoked TRPA1 response)
  99.27%
PF-04745637    
TRPA1, IC50: 17 nM
  98.65%
Olvanil  
TRPV1, EC50: 0.7 nM
    ≥99.0%
Capsiate  
TRPV1
    99.51%
MSP-3  
TRPV1, EC50: 0.87 μM
   
Methyl kakuol    
TRPA1
 
JTS-653  
TRPV1
   
TRPV1 antagonist 3  
hTRPV1, IC50: 2.66 nM
   
L-R4W2 TFA  
TRPV1, IC50: 0.1 μM
   
TRPV3 antagonist 74a  
TRPV3
   
L-R4W2  
TRPV1, IC50: 0.1 μM
   
D-erythro-Sphingosine hydrochloride
TRPM3
     
M8-B
TRPM8
     
Chrysin 6-C-glucoside 8-C-arabinoside  
TRPV1
   
Dihydrocapsiate  
TRPV1
    99.18%
AMG8788    
TRPA1, IC50: 1 μM
 
AMG9678    
TRPA1, IC50: 0.6 μM
 
N-Arachidonyldopamine  
TRPV1, EC50: ~50 nM
   
V116517  
TRPV1