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Results for "

CBZ

" in MedChemExpress (MCE) Product Catalog:

By Targets:	ADC Linker (10) Amino Acid Derivatives (11) Amyloid-β (1) Autophagy (5) Beta-lactamase (3) Biochemical Assay Reagents (23) Calcium Channel (2) Caspase (1) Cathepsin (3) Cholinesterase (ChE) (1) COX (1) DNA/RNA Synthesis (2) Drug Derivative (3) Drug Intermediate (9) Drug Isomer (1) Drug-Linker Conjugates for ADC (2) Factor Xa (2) Fluorescent Dye (6) Glutaminase (2) HDAC (2) HSV (1) Influenza Virus (1) Isotope-Labeled Compounds (6) Kallikrein (1) Liposome (1) Lipoxygenase (1) LYTACs (1) Microtubule/Tubulin (1) Mitophagy (5) MMP (1) mTOR (1) Nucleoside Antimetabolite/Analog (1) Phosphoramidites (1) Potassium Channel (2) PROTAC Linkers (44) PROTACs (1) Reference Standards (2) SARS-CoV (2) Ser/Thr Protease (3) Sodium Channel (5) Stearoyl-CoA Desaturase (SCD) (2) Thrombin (1)
By Research Areas:	Cancer (67) Cardiovascular Disease (2) Infection (7) Inflammation/Immunology (4) Metabolic Disease (1) Neurological Disease (10)
Click Chemistry:	Azide (1) Alkynes (1)
Oligonucleotides:	Cytosine (1) Phosphoramidites (1)

132

Inhibitors & Agonists

Fluorescent Dyes

Biochemical Assay Reagents

Peptides

Isotope-Labeled Compounds

Click Chemistry

Oligonucleotides

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-B0246

Carbamazepine Maximum Cited Publications 17 Publications Verification CBZ; NSC 169864	Sodium Channel Autophagy Mitophagy Potassium Channel Calcium Channel HDAC	Neurological Disease Cancer
Carbamazepine is an orally active pressure-sensitive sodium ion channel blocker with an IC₅₀ of 131 μM. Carbamazepine blocks voltage gated Na ⁺, Ca ²⁺, and K ⁺ channels, and is also a HDAC inhibitor (IC₅₀: 2 μM). Carbamazepine is an anticonvulsant and can be used for research of epilepsy and neuropathic pain .

HY-136626

Z-Ala-Ala-Asn-AMC 3 Publications Verification CBZ-Ala-Ala-Asn-AMC	Fluorescent Dye	Cancer
Z-Ala-Ala-Asn-AMC (Cbz-Ala-Ala-Asn-AMC) is the legumain substrate. Overexpressed legumain in 293 HEK-Leg cells potently cleaved CBZ-Ala-Ala-Asn-AMC .

HY-129126

NC9 1 Publications Verification CBZ-Lys(Acr)-PEG2-dansyl	Glutaminase Microtubule/Tubulin	Others
NC9 (Cbz-Lys(Acr)-PEG2-dansyl) is an irreversible transglutaminase (TG) inhibitor. NC9 inhibits osteoblast differentiation and mineralization. NC9 destabilizes microtubules. NC9 can be used for the research of osteoblast differentiation .

HY-P1759

*N-CBZ-Phe-Arg-AMC* Z-FR-AMC	Cathepsin	Others
N-CBZ-Phe-Arg-AMC (Z-FR-AMC) is a cathepsin substrate used in assessment activity of lysosomal cathepsin enzymes .

HY-B0246S

Carbamazepine-d10 CBZ-d₁₀; NSC 169864-d₁₀	Sodium Channel Autophagy Mitophagy	Neurological Disease Cancer
Carbamazepine-d₁₀ is the deuterium labeled Carbamazepine. Carbamazepine (CBZ), a sodium channel blocker, is an anticonvulsant agent .

HY-147354

TriGalNAc CBz	LYTACs	Cardiovascular Disease
TriGalNAc CBz is a GalNAc derivative and tri-GalNAc is an asialoglycoprotein receptor (ASGPR) ligand. TriGalNAc CBz can be used for mRNA drug delivery as well as lysosomal targeted chimerism (LYTAC) studies .

HY-W016042

*N-Cbz-Hydroxy-L-proline*	Drug Intermediate	Others
N-Cbz-Hydroxy-L-proline is a chiral N-Cbz-protected amino acid derivative. N-Cbz-Hydroxy-L-proline is commonly used in the synthesis of polypeptides and pharmaceutical intermediates. N-Cbz-Hydroxy-L-proline undergoes decarboxylation under AlCl₃/HFIP conditions .

HY-B0246R

Carbamazepine (Standard) CBZ (Standard); NSC 169864 (Standard)	Reference Standards Sodium Channel Autophagy Mitophagy Potassium Channel Calcium Channel HDAC	Neurological Disease Cancer
Carbamazepine (Standard) is the analytical standard of Carbamazepine. This product is intended for research and analytical applications. Carbamazepine is an orally active pressure-sensitive sodium ion channel blocker with an IC₅₀ of 131 μM. Carbamazepine blocks voltage gated Na ⁺, Ca ²⁺, and K ⁺ channels, and is also a HDAC inhibitor (IC₅₀: 2 μM). Carbamazepine is an anticonvulsant and can be used for research of epilepsy and neuropathic pain .

HY-P1759A

*N-CBZ-Phe-Arg-AMC hydrochloride* Z-FR-AMC hydrochloride	Cathepsin	Others
N-CBZ-Phe-Arg-AMC (Z-FR-AMC) hydrochloride is a cathepsin substrate used in assessment activity of lysosomal cathepsin enzymes .

HY-B0246S2

Carbamazepine-d8 CBZ-d₈; NSC 169864-d₈	Isotope-Labeled Compounds Sodium Channel Autophagy Mitophagy	Neurological Disease Cancer
Carbamazepine-d₈ is the deuterium labeled Carbamazepine. Carbamazepine, a sodium channel blocker, is an anticonvulsant agent, with an IC₅₀ of 131 μM .

HY-114267

Cbz-B3A	mTOR	Others
Cbz-B3A is a potent and selective inhibitor of mTORC1 signaling that appear to bind to ubiquilins 1, 2, and 4, and Cbz-B3A inhibits the phosphorylation of eIF4E-binding protein 1 (4EBP1).

HY-Y0588

Carbobenzoxyproline L-CBZ-Proline	MMP	Others
Carbobenzoxyproline (L-Cbz-Proline) is an inhibitor of prolidase. Carbobenzoxyproline can be used for prolidase deficiency (PD) research .

HY-W095029

Cbz-Gly-Pro-OH	Biochemical Assay Reagents	Others
Cbz-Gly-Pro-OH is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-W011750

Z-Pyr-OH CBZ-L-pyroglutamic acid	Biochemical Assay Reagents	Others
Z-Pyr-OH (Cbz-L-pyroglutamic acid) can be used as a biochemical assay reagent .

HY-45669

Fmoc-Gly-Gly-Phe-Gly-CH2-O-CH2-Cbz	PROTAC Linkers	Cancer
Fmoc-Gly-Gly-Phe-Gly-CH2-O-CH2-Cbz is a PROTAC linker and a maleimide-GGFG peptide linker. Fmoc-Gly-Gly-Phe-Gly-CH2-O-CH2-Cbz can be used in the synthesis of the Deruxtecan .

HY-W011197

Cbz-L-Trp-OH	Stearoyl-CoA Desaturase (SCD)	Inflammation/Immunology Cancer
Cbz-L-Trp-OH is a competitive inhibitor of SCD, with an IC₅₀ of 2.5 μM and a K_i of 2.1 μM .

HY-140488

Cbz-NH-PEG3-C2-acid	PROTAC Linkers	Cancer
Cbz-NH-PEG3-C2-acid is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-B0246S3

Carbamazepine-(Ph)d8 CBZ-(Ph)d₈; NSC 169864-(Ph)d₈	Isotope-Labeled Compounds	Neurological Disease Cancer
Carbamazepine-(Ph)d8 (CBZ-(Ph)d8; NSC 169864-(Ph)d8) is the deuterium labeled Carbamazepine-(Ph) (HY-B0246) .

HY-134113

Z-Gly-Pro-Arg-pNA CBZ-Chromozym TH	Biochemical Assay Reagents	Others
Z-Gly-Pro-Arg-pNA (z-GPR-pNA) is a photometric substrate in Prostate-Specific Antigen (PSA) activation protease assays. Z-Gly-Pro-Arg-pNA (z-GPR-pNA) can be used for the test of trypsin activity .

HY-177209

**Cbz-Val-(triAc-β-D-glucoside methyl ester)-Cbz**	Drug Intermediate	Cancer
Cbz-Val-(triAc-β-D-glucoside methyl ester)-Cbz is an intermediate used in the synthesis of ADC drug-linker .

HY-77475

*1-Cbz-3-Hydroxyazetidine*	ADC Linker PROTAC Linkers	Cancer
1-Cbz-3-Hydroxyazetidine is a non-cleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs). 1-Cbz-3-Hydroxyazetidine is also a alkyl chain-based PROTAC linker that can be used in the synthesis of PROTACs.

HY-78897

CBZ-L-Isoleucine	Amino Acid Derivatives	Others
CBZ-L-Isoleucine is an isoleucine derivative .

HY-P5027

Cbz-Lys-Arg-pNA	Ser/Thr Protease Kallikrein Factor Xa Thrombin	Cardiovascular Disease
Cbz-Lys-Arg-pNA is a peptide substrate containing pNA as the chromogenic group. Cbz-Lys-Arg-pNA is widely used in enzymatic analysis, including thrombin, plasmin, factor Xa and Kallikrein .

HY-W009503

Cbz-L-Aspartic anhydride	Amino Acid Derivatives	Others
Cbz-L-Aspartic anhydride is an aspartic acid derivative .

HY-46346

Fmoc-Gly-NH-CH2-O-CH2-Cbz	PROTAC Linkers	Cancer
Fmoc-Gly-NH-CH2-O-CH2-Cbz is a PROTAC linker and a maleimide-GGFG peptide linker. Fmoc-Gly-NH-CH2-O-CH2-Cbz can be used in the synthesis of the Deruxtecan .

HY-W025724

PEG2-NH-Cbz	PROTAC Linkers	Cancer
PEG2-NH-Cbz is a PROTAC linker that can be used in the synthesis of PROTACs.

HY-W004868

*1-Cbz-azetidine-3-carboxylic acid*	ADC Linker PROTAC Linkers	Cancer
1-Cbz-azetidine-3-carboxylic acid is a non-cleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs). 1-Cbz-azetidine-3-carboxylic acid is also a alkyl chain-based PROTAC linker that can be used in the synthesis of PROTACs[1]

HY-W336455

Cbz-PEG2-C2-NH2	PROTAC Linkers	Cancer
Cbz-PEG2-C2-NH2 is a PROTAC linker that can be used in the synthesis of PROTACs.

HY-B0246S4

Carbamazepine-d4 CBZ-d₄; NSC 169864-d₄	Isotope-Labeled Compounds	Others
Carbamazepine-d₄ (CBZ-d₄) is the deuterium labeled Carbamazepine (HY-B0246) . Carbamazepine is an orally active pressure-sensitive sodium ion channel blocker with an IC₅₀ of 131 μM. Carbamazepine blocks voltage gated Na ⁺, Ca ²⁺, and K ⁺ channels, and is also a HDAC inhibitor (IC₅₀: 2 μM). Carbamazepine is an anticonvulsant and can be used for research of epilepsy and neuropathic pain.

HY-B0246S1

Carbamazepine-d2 CBZ-d₂; NSC 169864-d₂	Isotope-Labeled Compounds Sodium Channel Autophagy Mitophagy	Neurological Disease Cancer
Carbamazepine-d₂ is the deuterium labeled Carbamazepine. Carbamazepine, a sodium channel blocker, is an anticonvulsant agent.

HY-160255

*N-Cbz-L-Cysteine* CBZ-cysteine	Beta-lactamase	Infection
N-Cbz-L-Cysteine (Cbz-cysteine) (compound 5) is a potent β-lactamase II inhibitor with a K_i value of 97 µM .

HY-W013905

Cbz-D-Valine	Amino Acid Derivatives	Others
Cbz-D-Valine is a valine derivative .

HY-W294220

*3-(Cbz-aminomethyl)azetidine hydrochloride*	PROTAC Linkers	Cancer
3-(Cbz-aminomethyl)azetidine (hydrochloride) is a PROTAC linker that can be used in the synthesis of PROTACs.

HY-W009121

Cbz-D-Trp-OH	Stearoyl-CoA Desaturase (SCD)	Inflammation/Immunology Cancer
Cbz-D-Trp-OH is a competitive inhibitor of SCD, with IC₅₀ of 86 μM and K_i of 71 μM .

HY-76317

Z-DL-Pro-OH N-CBZ-DL-proline; DL-CBZ-Proline	Amino Acid Derivatives	Others
Z-DL-Pro-OH (N-Cbz-DL-proline) is a proline derivative, can be used for the synthesis of agents or other compounds .

HY-W009033

Cbz-Lys(Boc)-OH	Biochemical Assay Reagents Amino Acid Derivatives	Others
Cbz-Lys(Boc)-OH is a protected amino acid, primarily utilized in peptide synthesis, protein engineering, and drug development, particularly in research involving lysine residues .

HY-W057967

Cbz-azaspiro[3.3]heptane-OH	PROTAC Linkers	Cancer
Cbz-azaspiro[3.3]heptane-OH is a PROTAC linker that can be used in the synthesis of PROTACs.

HY-133358

Cbz-NH-PEG12-C2-acid	PROTAC Linkers	Cancer
Cbz-NH-PEG12-C2-acid is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-130192

Cbz-NH-PEG8-C2-acid	PROTAC Linkers	Cancer
Cbz-NH-PEG8-C2-acid is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-140487

Cbz-NH-PEG2-C2-acid	PROTAC Linkers	Cancer
Cbz-NH-PEG2-C2-acid is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-140489

Cbz-NH-PEG5-C2-acid	PROTAC Linkers	Cancer
Cbz-NH-PEG5-C2-acid is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-135925

Cbz-NH-PEG1-CH2COOH	PROTAC Linkers	Cancer
Cbz-NH-PEG1-CH2COOH is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-135923

Cbz-NH-PEG2-CH2COOH	PROTAC Linkers	Cancer
Cbz-NH-PEG2-CH2COOH is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-135913

Cbz-NH-PEG3-CH2COOH	PROTAC Linkers	Cancer
Cbz-NH-PEG3-CH2COOH is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-135926

Cbz-NH-PEG1-CH2CH2COOH	PROTAC Linkers	Cancer
Cbz-NH-PEG1-CH2CH2COOH is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs .

HY-P10198

Cbz-Lys-Lys-PABA-AMC diTFA	Fluorescent Dye	Others
Cbz-Lys-Lys-PABA-AMC diTFA is a fluorogenic peptide .

HY-W103577

*1-(Cbz-amino)cyclopentanecarboxylic acid* CBZ-cycloleucine	Biochemical Assay Reagents	Others
1-(Cbz-amino)cyclopentanecarboxylic acid (Cbz-cycloleucine) is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-160255A

*N-Cbz-D-Cysteine* CBZ-D-Cys	Beta-lactamase	Infection
N-Cbz-D-Cysteine (Cbz-D-Cys) (compound 5) is a potent β-lactamase II inhibitor with a K_i value of 20.1 µM .

HY-I1061

Cbz-L-Alloisoleucine	Amino Acid Derivatives	Others
Cbz-L-Alloisoleucine is an isoleucine derivative .

HY-126375R

Cbz-?Valaciclovir (Standard) Benzyloxycarbonyl valacyclovir (Standard)	Drug Intermediate Reference Standards	Infection
Cbz-Valaciclovir (Standard) is the analytical standard of Cbz-Valaciclovir. This product is intended for research and analytical applications. Cbz-Valaciclovir (Benzyloxycarbonyl valacyclovir) can be used to prepare Valaciclovir (HY-17425) and for antiviral research .

Cat. No.	Product Name	Type

HY-W016042

*N-Cbz-Hydroxy-L-proline*	Biochemical Assay Reagents
N-Cbz-Hydroxy-L-proline is a chiral N-Cbz-protected amino acid derivative. N-Cbz-Hydroxy-L-proline is commonly used in the synthesis of polypeptides and pharmaceutical intermediates. N-Cbz-Hydroxy-L-proline undergoes decarboxylation under AlCl₃/HFIP conditions .

HY-32685

*N-Cbz-1,2,3,6-tetrahydropyridine-4-boronic acid pinacol ester*	Biochemical Assay Reagents
N-Cbz-1,2,3,6-tetrahydropyridine-4-boronic acid pinacol ester is a biochemical reagent.

HY-P1759A

*N-CBZ-Phe-Arg-AMC hydrochloride* Z-FR-AMC hydrochloride	Biochemical Assay Reagents
N-CBZ-Phe-Arg-AMC (Z-FR-AMC) hydrochloride is a cathepsin substrate used in assessment activity of lysosomal cathepsin enzymes .

HY-W008753

Z-L-Val-OH N-CBZ-L-valine	Biochemical Assay Reagents
Z-L-Val-OH (N-Cbz-L-valine) is an amino acid derivative and key intermediate in organic synthesis. Z-L-Val-OH can be used in the synthesis of anti-cytomegalovirus compounds and peptide inhibitors of human spleen plasminogen activator (SFP) and human leukocyte elastase-like protease (ELP) .

HY-W402032

*Bis-Cbz-cyclen*	Biochemical Assay Reagents
Bis-Cbz-cyclen is a bifunctional chelator. Bifunctional chelating agents are used to stably link the radiometal to the carrier moiety of the radiopharmaceutical .

Cat. No.	Product Name	Target	Research Area

HY-136626

Z-Ala-Ala-Asn-AMC 3 Publications Verification CBZ-Ala-Ala-Asn-AMC	Fluorescent Dye	Cancer
Z-Ala-Ala-Asn-AMC (Cbz-Ala-Ala-Asn-AMC) is the legumain substrate. Overexpressed legumain in 293 HEK-Leg cells potently cleaved CBZ-Ala-Ala-Asn-AMC .

HY-P1759

*N-CBZ-Phe-Arg-AMC* Z-FR-AMC	Cathepsin	Others
N-CBZ-Phe-Arg-AMC (Z-FR-AMC) is a cathepsin substrate used in assessment activity of lysosomal cathepsin enzymes .

HY-P1759B

*N-CBZ-Phe-Arg-AMC TFA* Z-FR-AMC TFA	Cathepsin	Others
N-CBZ-Phe-Arg-AMC (Z-FR-AMC) TFA is a cathepsin substrate used in assessment activity of lysosomal cathepsin enzymes .

HY-W011750

Z-Pyr-OH CBZ-L-pyroglutamic acid	Biochemical Assay Reagents	Others
Z-Pyr-OH (Cbz-L-pyroglutamic acid) can be used as a biochemical assay reagent .

HY-134113

Z-Gly-Pro-Arg-pNA CBZ-Chromozym TH	Biochemical Assay Reagents	Others
Z-Gly-Pro-Arg-pNA (z-GPR-pNA) is a photometric substrate in Prostate-Specific Antigen (PSA) activation protease assays. Z-Gly-Pro-Arg-pNA (z-GPR-pNA) can be used for the test of trypsin activity .

HY-P3106

(Z-Ala-Ala-Ala-Ala)2Rh110 (Z-Ala-Ala-Ala-Ala)2Rhodamine110; bis-CBZ-L-alanyl-L-arginine amide Rhodamine 110	Fluorescent Dye	Others
(Z-Ala-Ala-Ala-Ala)2Rh110 is a sensitive fluorogenic elastase substrate. The colorless and nonfluorescent (Z-Ala-Ala-Ala-Ala)2Rh110 is selectively cleaved by elastase to yield the highly fluorescent compound rhodamine 110, which can be analyzed with an excitation wavelength of 485 nm and emission wavelength of 525 nm.

HY-78897

CBZ-L-Isoleucine	Amino Acid Derivatives	Others
CBZ-L-Isoleucine is an isoleucine derivative .

HY-P5027

Cbz-Lys-Arg-pNA	Ser/Thr Protease Kallikrein Factor Xa Thrombin	Cardiovascular Disease
Cbz-Lys-Arg-pNA is a peptide substrate containing pNA as the chromogenic group. Cbz-Lys-Arg-pNA is widely used in enzymatic analysis, including thrombin, plasmin, factor Xa and Kallikrein .

HY-W009503

Cbz-L-Aspartic anhydride	Amino Acid Derivatives	Others
Cbz-L-Aspartic anhydride is an aspartic acid derivative .

HY-P5042

Cbz-Tyr-Ala-OH	Peptides	Others
Cbz-Tyr-Ala-OH is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development .

HY-W003991

*N-Benzyl-N-Cbz-glycine*	Amino Acid Derivatives	Others
2-(Benzyl(tert-butoxycarbonyl)amino)acetic acid is a Glycine (HY-Y0966) derivative .

HY-W013905

Cbz-D-Valine	Amino Acid Derivatives	Others
Cbz-D-Valine is a valine derivative .

HY-76317

Z-DL-Pro-OH N-CBZ-DL-proline; DL-CBZ-Proline	Amino Acid Derivatives	Others
Z-DL-Pro-OH (N-Cbz-DL-proline) is a proline derivative, can be used for the synthesis of agents or other compounds .

HY-75332

Z-D-Phg-OH D-CBZ phenylglycine	Amino Acid Derivatives	Others
Z-D-Phg-OH (D-Cbz phenylglycine) is a N-blocked amino acids with K_d values of 390 μM and 323 μM for tBuCQN and tBuCQD, respectively .

HY-P5024

Cbz-Ile-Pro-OH NSC 333754	Peptides	Others
Cbz-Ile-Pro-OH (NSC 333754) is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development .

HY-P10198

Cbz-Lys-Lys-PABA-AMC diTFA	Fluorescent Dye	Others
Cbz-Lys-Lys-PABA-AMC diTFA is a fluorogenic peptide .

HY-I1061

Cbz-L-Alloisoleucine	Amino Acid Derivatives	Others
Cbz-L-Alloisoleucine is an isoleucine derivative .

HY-400312

Cbz-D-Leu-Val-Boc	Biochemical Assay Reagents	Cancer
Cbz-D-Leu-Val-Boc is a peptide derivative.

HY-P5040

Cbz-Pro-Leu-Gly-OH	Peptides	Neurological Disease
Cbz-Pro-Leu-Gly-OH is a tripeptide that can be used in Parkinson's disease research .

HY-P5008

Cbz-Asn-Gly-OH CBZ-Asn-Gly; Z-Asn-Gly-OH	Peptides	Others
Cbz-Asn-Gly-OH is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development .

HY-P5012

Cbz-Glu-Gly-OH NSC 186902	Peptides	Others
Cbz-Glu-Gly-OH (NSC 186902) is a polypeptide that can be found by peptide screening. Peptide screening is a research tool that pools active peptides primarily by immunoassay. Peptide screening can be used for protein interaction, functional analysis, epitope screening, especially in the field of agent research and development .

HY-173459

N-0920	SARS-CoV	Infection
N-0920 is a potent TMPRSS2 inhibitor with an IC₅₀ of 0.35 nM. N-0920 effectively inhibits SARS-CoV-2 variants EG.5.1 and JN.1 entry in Calu-3 cells, with picomolar EC₅₀s values of 300 pM and 90 pM, respectively .

HY-P10213

CbZ-Ala-Ala-Ala-Ala	Peptides	Others
CbZ-Ala-Ala-Ala-Ala is a modified peptide .

HY-P2269A

MAIT-203 acetate	Drug Derivative	Cancer
MAIT-203 acetate is a cyclopentyalanin-derived peptidomimetic, potently inhibits the interaction of adenomatous polyposis coli (APC) and Asef (RhoGEF4), but not APC-Sam68 or APC-striatin interactions. MAIT-203 acetate binds APC-ARM with a K_i value of 0.015 μM and aK_d value of 0.036 μM. MAIT-203 acetate significantly represses the migration and invasion of colorectal cancer cells .

HY-P2269

MAIT-203	Drug Derivative	Cancer
MAIT-203, a cyclopentyalanin-derived peptidomimetic, potently inhibits the interaction of adenomatous polyposis coli (APC) and Asef (RhoGEF4), but not APC-Sam68 or APC-striatin interactions. MAIT-203 binds APC-ARM with a K_i of 0.015 μM and a K_d of 0.036 μM. MAIT-203 significantly represses the migration and invasion of colorectal cancer cells.

HY-W060779

*(4R)-1-Cbz-4-hydroxy-D-proline methyl ester*	Amino Acid Derivatives	Others
1-Benzyl 2-methyl (2R,4R)-4-hydroxypyrrolidine-1,2-dicarboxylate is a proline derivative .

HY-P11476

(Z-AR)2Rh110	Ser/Thr Protease Fluorescent Dye Drug Derivative	Others
(Z-AR)2Rh110 is a Rhodamine derivative. (Z-AR)2Rh110 can be hydrolyzed by trypsin .

HY-D3169

IETDC	Fluorescent Dye Caspase	Inflammation/Immunology
IETDC is a caspase 8 probe substrate. IETDC is cleaved by activated caspase 8 to release D-cysteine. The D-cysteine released by IETDC binds to HCBT to generate firefly luciferin in situ, accompanied by a bioluminescent signal produced by H₂O₂-mediated release of 6-hydroxy-2-cyanobenzothiazole. IETDC is applicable to studies related to acute inflammation .

Cat. No.	Product Name	Chemical Structure

HY-B0246S

Carbamazepine-d10
Carbamazepine-d₁₀ is the deuterium labeled Carbamazepine. Carbamazepine (CBZ), a sodium channel blocker, is an anticonvulsant agent .

HY-B0246S2

Carbamazepine-d8
Carbamazepine-d₈ is the deuterium labeled Carbamazepine. Carbamazepine, a sodium channel blocker, is an anticonvulsant agent, with an IC₅₀ of 131 μM .

HY-B0246S3

Carbamazepine-(Ph)d8
Carbamazepine-(Ph)d8 (CBZ-(Ph)d8; NSC 169864-(Ph)d8) is the deuterium labeled Carbamazepine-(Ph) (HY-B0246) .

HY-B0246S4

Carbamazepine-d4

Carbamazepine-d₄ (CBZ-d₄) is the deuterium labeled Carbamazepine (HY-B0246) . Carbamazepine is an orally active pressure-sensitive sodium ion channel blocker with an IC₅₀ of 131 μM. Carbamazepine blocks voltage gated Na ⁺, Ca ²⁺, and K ⁺ channels, and is also a HDAC inhibitor (IC₅₀: 2 μM). Carbamazepine is an anticonvulsant and can be used for research of epilepsy and neuropathic pain.

HY-B0246S1

Carbamazepine-d2
Carbamazepine-d₂ is the deuterium labeled Carbamazepine. Carbamazepine, a sodium channel blocker, is an anticonvulsant agent.

HY-W777099

*N-Cbz-O-Bzl-L-Glu-S-Bzl-L-Cys-Gly[13C2,15N]-OBzl*
N-Cbz-O-Bzl-L-Glu-S-Bzl-L-Cys-Gly[ ¹³C₂, ¹⁵N]-OBzl is the ¹³C- and ¹⁵N-labeled N-Cbz-O-Bzl-L-Glu-S-Bzl-L-Cys-Gly-OBzl.

HY-W653882

Carbamazepine-d2,15N
Carbamazepine-d2,15N is a deuterated labeled Carbamazepine-d2,15N .

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