70 Results for "

Tyr-Gly-Gly

" in MedChemExpress (MCE) Product Catalog:
Products (70)

70 Results for "Tyr-Gly-Gly" in MCE Product Catalog:

37
37 Publications Verification
Cat. No.: HY-P0017
CAS No.: 9087-70-1
Aprotinin is a bovine pancreatic trypsin inhibitor (BPTI) inhibitor which inhibits trypsin and chymotrypsin with Kis of 0.06 pM and 9 nM, respectively.
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4
4 Cited Publications
Cat. No.: HY-P0073
CAS No.: 58569-55-4
Synonyms: Met-Enkephalin; Methionine enkephalin; Metenkefalin
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease Cancer

Tyr-Gly-Gly-Phe-Met-OH regulates human immune function and inhibits tumor growth via binding to the opioid receptor.
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3
3 Cited Publications
Cat. No.: HY-P2341
Target:  

LDLR

Research Areas:  

Cancer

Angiopep-2 hydrochloride is a brain peptide vector. The conjugation of anticancer agents with the Angiopep-2 peptide vector could increase their efficacy in the treatment of brain cancer .
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2
2 Cited Publications
Cat. No.: HY-P0288
CAS No.: 58822-25-6
Synonyms: Leu-enkephalin; Leucine enkephalin; Leucyl-enkephalin
[Leu5]-Enkephalin is a pentapeptide with morphine like properties. [Leu5]-Enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.
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2
2 Cited Publications
Cat. No.: HY-P1333
CAS No.: 80448-90-4
Dynorphin A is an endogenous opioid peptide involved in inhibitory neurotransmission in the central nervous system (CNS). Dynorphin A is a highy potent kappa opioid receptor (KOR) agonist, and is also an agonist for other opioid receptors, such as mu (MOR) and delta (DOR). Dynorphin A can induce neuronal death, and can be used in the research of neurological disease .
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2
2 Cited Publications
Cat. No.: HY-108814A
Purity:  97.69%
Synonyms: DX-88 TFA
Target:  

Kallikrein

Research Areas:  

Cardiovascular Disease

Ecallantide (DX-88) TFA is a specific recombinant plasma kallikrein inhibitor. Ecallantide inhibits the production of bradykinin. Ecallantide may be used to prevent acute attacks of angioedema .
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1
1 Cited Publications
Cat. No.: HY-P1502
CAS No.: 61214-51-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus, is an agonist of opioid receptor, with preferred affinity for μ-opioid receptor and δ-opioid receptor; β-Endorphin, human exhibits antinociception activity.
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1
1 Cited Publications
Cat. No.: HY-P10908
CAS No.: 3020015-02-2
Target:  

PD-1/PD-L1

Research Areas:  

Others

H-20 is a PD-1 agonist. H-20 can be used in the research of chronic pain .
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1
1 Cited Publications
Cat. No.: HY-P1337
CAS No.: 83335-41-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.
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1
1 Cited Publications
Cat. No.: HY-P1337A
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor.
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1
1 Cited Publications
Cat. No.: HY-P1866A
β-Endorphin, equine TFA is an endogenous opioid peptide, which binds at high affinity to both μ/δ opioid receptors. β-Endorphin, equine TFA has analgesic properties .
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1
1 Cited Publications
Cat. No.: HY-P4106A
Research Areas:  

Neurological Disease

Tat-GluR23Y, scrambled TFA is the scrambled peptide of Tat-GluR23Y (HY-P2259). Tat-GluR23Y is a synthetic peptide containing tyrosine residues that inhibit AMPAR endocytosis and is effective in the research of long-term depression (LTD) .
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Cat. No.: HY-P1351
CAS No.: 906480-09-9
Research Areas:  

Cancer

Angiopep-2-cys is a conjugate of Angiopep-2 hydrochloride (HY-P2341) and cysteine. Angiopep-2 hydrochloride is a brain peptide vector. The conjugation of anticancer agents with the Angiopep-2 peptide vector could increase their efficacy in the treatment of brain cancer .
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Cat. No.: HY-P4073
CAS No.: 1075214-55-9
Synonyms: GRN1005; Paclitaxel trevatide
Research Areas:  

Cancer

ANG1005 (Paclitaxel trevatide) is a brain-penetrating peptide-drug conjugate. ANG1005, a taxane derivative, consists of three paclitaxel (HY-B0015) molecules covalently linked to Angiopep-2, designed to cross the blood-brain and blood-cerebrospinal barriers and to penetrate malignant cells via low density lipoprotein receptor-related protein (LRP1) transport system .
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Cat. No.: HY-P2159
CAS No.: 75790-53-3
Dynorphin A (1-8) is a ligand with preference for the κ-opioid receptor, and its IC50 value against human placental κ-opioid receptor is 330 nM. Dynorphin A (1-8) mediates neuroprotective effects by inhibiting oxidative stress, suppressing apoptosis, and competitively displacing the binding of κ partial agonists. Dynorphin A (1-8) is the dominant opioid peptide in human placental villi and tissue extracts; it undergoes rapid hydrolysis and can enter the central nervous system via intranasal administration. Dynorphin A (1-8) can be used in studies related to ischemic stroke .
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Cat. No.: HY-P1087
CAS No.: 88377-68-8
Synonyms: Metorphamide
Target:  

Opioid Receptor

Research Areas:  

Cancer

Adrenorphin is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM.
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Cat. No.: HY-P0088
CAS No.: 72957-38-1
Synonyms: Dynorphin A Porcine Fragment 1-13
Target:  

Opioid Receptor

Research Areas:  

Others

Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations.
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Cat. No.: HY-P1470
CAS No.: 60117-24-0
Synonyms: Leu-Enkephalin amide
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

[Leu5]-Enkephalin, amide is a δ opioid receptor agonist.
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Cat. No.: HY-P11195
Target:  

Drug Derivative

Research Areas:  

Neurological Disease

Angiopep-2 azide is a peptide derivative of Angiopep-2 (HY-P2341) bearing a side chain azide (N3) group. Angiopep-2 exhibits high blood-brain barrier (BBB) penetration capability and can be used for brain compound delivery .
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Cat. No.: HY-P1170
CAS No.: 2703746-32-9
Synonyms: Ac-L-Tyr-Gly-Gly-L-Phe-D-Leu-COOH
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

N-terminally acetylated Leu-enkephalin is the N-terminally acetylated form of Leu-enkephalin. Leu-enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.
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