1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor

Adrenorphin (Synonyms: Metorphamide)

Cat. No.: HY-P1087 Purity: 95.49%
Handling Instructions

Adrenorphin is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM. Sequence: Tyr-Gly-Gly-Phe-Met-Arg-Arg-Val-NH2;YGGFMRRV-NH2.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

Adrenorphin Chemical Structure

Adrenorphin Chemical Structure

CAS No. : 88377-68-8

Size Price Stock Quantity
1 mg USD 70 In-stock
Estimated Time of Arrival: December 31
5 mg USD 210 In-stock
Estimated Time of Arrival: December 31
10 mg   Get quote  
50 mg   Get quote  

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Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Adrenorphin is a opioid octapeptide, acting as a potent agonist of μ-opioid receptor, with Ki of 12 nM. Sequence: Tyr-Gly-Gly-Phe-Met-Arg-Arg-Val-NH2;YGGFMRRV-NH2.

IC50 & Target

Ki: 12 nM (μ-opioid receptor)[1]

In Vitro

Adrenorphin (Metorphamide) is a opioid octapeptide from bovine brain, acts as a potent agonist of μ-opioid receptor, with Ki of 12 nM. The binding ratios of Ki for μ-opioid receptor/Ki for δ-opioid receptor of 0.04 and of Ki for μ-opioid receptor/Ki for κ-opioid receptor of 0.46[1]. Adrenorphin potently inhibits catecholamine secretion evoked by 10 μM nicotine in cultured human pheochromocytoma 6 cells, with an IC50 of 1.1 μM[2].

Solvent & Solubility
In Vitro: 

10 mM in H2O

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.0161 mL 5.0804 mL 10.1607 mL
5 mM 0.2032 mL 1.0161 mL 2.0321 mL
10 mM 0.1016 mL 0.5080 mL 1.0161 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

984.18

Formula

C₄₄H₆₉N₁₅O₉S

CAS No.

88377-68-8

Storage
Powder -80°C 2 years
  -20°C 1 year
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Adrenorphin
Cat. No.:
HY-P1087
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Adrenorphin

Cat. No.: HY-P1087