1. Signaling Pathways
  2. Antibody-drug Conjugate/ADC Related
  3. Drug-Linker Conjugates for ADC
  4. Drug-Linker Conjugates for ADC Inhibitors

Drug-Linker Conjugates for ADC Inhibitors

Auristatin

Camptothecins

Daunorubicins/Doxorubicins

Duocarmycins

Maytansinoids

Pyrrolobenzodiazepines

Traditional Cytotoxic Agents

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Drug-Linker Conjugates for ADC Inhibitors & Chemicals
Product Name Auristatin Camptothecins Daunorubicins/Doxorubicins Duocarmycins Maytansinoids Pyrrolobenzodiazepines Traditional Cytotoxic Agents Purity
VcMMAE
Auristatin
            99.97%
Deruxtecan  
Camptothecins
          99.94%
CL2A-SN-38  
Camptothecins
          99.07%
Val-Cit-PAB-MMAE
Auristatin
            99.83%
Vipivotide tetraxetan            
Traditional Cytotoxic Agents
99.57%
SMCC-DM1        
Maytansinoids
    98.53%
McMMAF
Auristatin
            99.53%
MC-Val-Cit-PAB-MMAF
Auristatin
            98.16%
MC-GGFG-Exatecan  
Camptothecins
          99.71%
Tesirine          
Pyrrolobenzodiazepines
  98.10%
MC-Val-Cit-PAB-Exatecan  
Camptothecins
          99.55%
Mal-VC-PAB-DM1        
Maytansinoids
    99.12%
SPDB-DM4        
Maytansinoids
    99.91%
DBCO-PEG4-VC-PAB-MMAE      
Duocarmycins
      99.88%
MC-VA-PAB-Exatecan  
Camptothecins
          99.58%
DBCO-PEG4-GGFG-Dxd            
Traditional Cytotoxic Agents
98.64%
Doxorubicin-SMCC    
Daunorubicins/Doxorubicins
        98.80%
sulfo-SPDB-DM4        
Maytansinoids
    99.77%
CL2-SN-38  
Camptothecins
          99.78%
Vc-seco-DUBA      
Duocarmycins
      99.95%
Mc-MMAE
Auristatin
            99.38%
SGD-1910          
Pyrrolobenzodiazepines
 
Gly3-VC-PAB-MMAE
Auristatin
            99.63%
MC-VA-PABC-MMAE
Auristatin
            99.88%
MC-betaglucuronide-MMAE-1
Auristatin
            99.72%
Mal-PEG2-VCP-Eribulin            
Traditional Cytotoxic Agents
99.82%
SuO-Val-Cit-PAB-MMAE
Auristatin
            99.24%
MAL-di-EG-Val-Cit-PAB-MMAE
Auristatin
            98.04%
DBCO-PEG4-Val-Cit-PAB-MMAF
Auristatin
            99.99%
Mal-PEG8-Val-Cit-PAB-MMAE
Auristatin
            99.67%
MC-VC-PABC-Aur0101
Auristatin
            99.66%
MC-Val-Cit-PAB-duocarmycin chloride      
Duocarmycins
      98.16%
PEG4-aminooxy-MMAF
Auristatin
            99.83%
DBCO-PEG4-VA-PBD            
Traditional Cytotoxic Agents
MMAE-SMCC
Auristatin
            99.56%
DBCO-(PEG)3-VC-PAB-MMAE
Auristatin
           
N3-PEG3-vc-PAB-MMAE
Auristatin
            98.56%
MAC glucuronide phenol-linked SN-38  
Camptothecins
          98.01%
Lys-SMCC-DM1        
Maytansinoids
    99.61%
DBCO-(PEG2-VC-PAB-MMAE)2
Auristatin
            98.73%
(Rac)-Lys-SMCC-DM1        
Maytansinoids
    98.18%
SC-VC-PAB-MMAE
Auristatin
            99.29%
Azide-PEG4-VC-PAB-Doxorubicin    
Daunorubicins/Doxorubicins
        98.47%
MC-DOXHZN hydrochloride    
Daunorubicins/Doxorubicins
        ≥98.0%
SuO-Glu-Val-Cit-PAB-MMAE
Auristatin
            99.20%
DBM-MMAF
Auristatin
            99.74%
MC-Val-Cit-PAB-carfilzomib iodide            
Traditional Cytotoxic Agents
DBCO-PEG4-VC-PAB-DMEA-PNU-159682      
Duocarmycins
     
MC-VC-PABC-DNA31            
Traditional Cytotoxic Agents
98.71%
SPP-DM1        
Maytansinoids
   
MC-DM1        
Maytansinoids
   
MC-Val-Cit-PAB-Auristatin E
Auristatin
           
Mal-PEG4-VA-PBD          
Pyrrolobenzodiazepines
 
MC-Val-Cit-PAB-vinblastine            
Traditional Cytotoxic Agents
DM4-SMCC        
Maytansinoids
   
Vc-MMAD
Auristatin
            99.96%
Val-Cit-PAB-MMAF sodium
Auristatin
            98.43%
NAMPT inhibitor-linker 1            
Traditional Cytotoxic Agents
98.08%
Mal-Phe-C4-VC-PAB-MMAE
Auristatin
            99.30%
MC-Gly-Gly-Phe-Gly-Cyclobutanecarboxylic-Exatecan  
Camptothecins
          98.66%
Aminobenzenesulfonic auristatin E TFA
Auristatin
            99.39%
AcLys-PABC-VC-Aur0101
Auristatin
            98.49%
Ac-Lys-Val-Cit-PABC-MMAE
Auristatin
            99.99%
DBCO-PEG4-MMAF
Auristatin
           
Fmoc-Val-Cit-PAB-MMAE
Auristatin
           
Mal-C6-α-Amanitin    
Daunorubicins/Doxorubicins
        98.48%
NAMPT inhibitor-linker 2            
Traditional Cytotoxic Agents
98.11%
MAL-di-EG-Val-Cit-PAB-MMAF
Auristatin
            98.56%
PSMA-ALB-56            
Traditional Cytotoxic Agents
98.92%
Cys-mcMMAD
Auristatin
            98.77%
DM1-PEG4-DBCO        
Maytansinoids
    98.04%
Fmoc-Val-Cit-PAB-Duocarmycin TM      
Duocarmycins
      ≥99.0%
DGN549-C            
Traditional Cytotoxic Agents
MC-Val-Cit-PAB-rifabutin            
Traditional Cytotoxic Agents
MC-Val-Cit-PAB-Retapamulin            
Traditional Cytotoxic Agents
99.00%
MC-Val-Cit-PAB-Indibulin            
Traditional Cytotoxic Agents
MC-GGFG-(7ethanol-10NH2-11F-Camptothecin)  
Camptothecins
         
MC-Val-Cit-PAB-clindamycin            
Traditional Cytotoxic Agents
99.99%
Aminobenzenesulfonic auristatin E
Auristatin
           
Mc-Dexamethasone        
Maytansinoids
   
Mal-PEG4-VC-PAB-DMEA-Seco-Duocarmycin SA      
Duocarmycins
     
Mc-MMAD
Auristatin
            98.50%
MC-DOXHZN    
Daunorubicins/Doxorubicins
       
AcLysValCit-PABC-DMAE-SW-163D            
Traditional Cytotoxic Agents
Vat-Cit-PAB-Monomethyl Dolastatin 10
Auristatin
           
MC-VC-PAB-MMAD
Auristatin
           
TLR7/8 agonist 4 hydroxy-PEG10-acid            
Traditional Cytotoxic Agents
VCP-Eribulin            
Traditional Cytotoxic Agents
DBCO-PEG4-Ahx-DM1        
Maytansinoids
   
ST8155AA1            
Traditional Cytotoxic Agents
HS-(CH2)3CO-L-Ala-D-Ala-L-Ala-NH-CH2-S-(CH2)5-CO-DM        
Maytansinoids
   
TLR7/8 agonist 4 hydroxy-PEG10-acid hydrochloride            
Traditional Cytotoxic Agents
Nitro-PDS-Tubulysin M
Auristatin
           
Sulfo-PDBA-DM4        
Maytansinoids
   
MC-Sq-Cit-PAB-Gefitinib            
Traditional Cytotoxic Agents
MC-Val-Cit-PAB-dimethylDNA31            
Traditional Cytotoxic Agents
DM4-SPDP        
Maytansinoids
   
Val-Cit-PAB-MMAF
Auristatin
           
MC-VC-PABC-C6-alpha-Amanitin    
Daunorubicins/Doxorubicins
       
PSMA-Val-Cit-PAB-MMAE
Auristatin
           
N3-PEG8-Phe-Lys-PABC-Gefitinib            
Traditional Cytotoxic Agents
MB-VC-MGBA      
Duocarmycins
     
Sulfo-SPDB-DGN462        
Maytansinoids
   
DBA-DM4        
Maytansinoids
   
Rha-PEG3-SMCC            
Traditional Cytotoxic Agents
Aminooxy CatB-LXR            
Traditional Cytotoxic Agents
MAC glucuronide α-hydroxy lactone-linked SN-38  
Camptothecins
         
AmPEG6C2-Aur0131            
Traditional Cytotoxic Agents
MCC-Modified Daunorubicinol    
Daunorubicins/Doxorubicins
       
MC-VC-PAB-Tubulysin M
Auristatin
           
MC-Gly-Gly-Phe-Gly-amide-cyclopropanol-amide-Exatecan
Auristatin
           
MC-betaglucuronide-MMAE-2
Auristatin
           
OSu-Glu-VC-PAB-MMAD
Auristatin
           
MC-Sq-Cit-PAB-Dolastatin10
Auristatin
           
Lys-Nε-SPDB-DM4        
Maytansinoids
   
ST8154AA1            
Traditional Cytotoxic Agents
MC-VC(S)-PABQ-Tubulysin M
Auristatin
           
Mipsagargin            
Traditional Cytotoxic Agents
Desmethyl Vc-seco-DUBA      
Duocarmycins
     
MC-Alkyl-Hydrazine Modified MMAF
Auristatin
           
MP-PEG8-Val-Lys-Gly-7-MAD-MDCPT  
Camptothecins