1 Result for "

ASP 8062

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "ASP 8062" in MCE Product Catalog:

Cat. No.: HY-184060
CAS No.: 1704716-36-8
Target:  

GABA Receptor

Research Areas:  

Neurological Disease

ASP8062 is an orally active, blood-brain barrier-permeable selective GABAB receptor allosteric modulator. ASP8062 enhances GABA-mediated activation of GABAB receptors and strengthens GABAergic neurotransmission. ASP8062 reverses Reserpine (HY-N0480)-induced myalgia, regulates the sleep-wake cycle, increases delta wave power during non-REM sleep, and impairs motor coordination at high doses. ASP8062 penetrates the central nervous system with a half-life of 40-50 h. ASP8062 can be used in research related to opioid use disorder, fibromyalgia, chronic pain, and alcohol use disorder [1][2] [3][4].