2 Results for "

ASP8062

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "ASP8062" in MCE Product Catalog:

Cat. No.: HY-184060
CAS No.: 1704716-36-8
Target:  

GABA Receptor

Domaines de recherche:  

Neurological Disease

ASP8062 is an orally active, blood-brain barrier-permeable selective GABAB receptor allosteric modulator. ASP8062 enhances GABA-mediated activation of GABAB receptors and strengthens GABAergic neurotransmission. ASP8062 reverses Reserpine (HY-N0480)-induced myalgia, regulates the sleep-wake cycle, increases delta wave power during non-REM sleep, and impairs motor coordination at high doses. ASP8062 penetrates the central nervous system with a half-life of 40-50 h. ASP8062 can be used in research related to opioid use disorder, fibromyalgia, chronic pain, and alcohol use disorder [1][2] [3][4].
Cat. No.: HY-P10278
CAS No.: 133658-45-4
Target:  

Peptides

Domaines de recherche:  

Endocrinology

Anantin binds competitively to the receptor of atrial natriuretic factor (ANF) from bovine adrenal cortex (Kd = 0.6 μM) and acts as natriuretic peptide receptor A antagonist .