126 Results for "

CYS1

" in MedChemExpress (MCE) Product Catalog:
Products (126)

126 Results for "CYS1" in MCE Product Catalog:

11
11 Cited Publications
Art. -Nr.: HY-P0256
CAS. Nr.: 24345-16-2
Synonyms: Apamine
Apamin (Apamine) is an 18 amino acid peptide neurotoxin found in apitoxin (bee venom), is known as a specifically selective blocker of Ca 2+-activated K + (SK) channels and exhibits anti-inflammatory and anti-fibrotic activity [1].
11
11 Cited Publications
Art. -Nr.: HY-P0256A
Synonyms: Apamine TFA
Apamin TFA (Apamine TFA) is an 18 amino acid peptide neurotoxin found in apitoxin (bee venom), is known as a specifically selective blocker of Ca 2+-activated K + (SK) channels and exhibits anti-inflammatory and anti-fibrotic activity [1].
10
10 Cited Publications
Art. -Nr.: HY-P0049
CAS. Nr.: 113-79-1
Synonyms: Arg8-vasopressin; AVP
Target:  

Vasopressin Receptor

Forschungsgebiete:  

Neurological Disease Cancer

Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1.
10
10 Cited Publications
Art. -Nr.: HY-W539944
CAS. Nr.: 129979-57-3
Synonyms: Arg8-vasopressin acetate; AVP acetate
Forschungsgebiete:  

Neurological Disease Cancer

Argipressin (Arg8-vasopressin) (acetate) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1 [1] .
9
9 Cited Publications
Art. -Nr.: HY-P0202
CAS. Nr.: 117399-94-7
Synonyms: ET-1 (swine, human)
Endothelin 1 (swine, human) (ET-1) is a synthetic peptide with the sequence of human and swine Endothelin 1, which is a potent endogenous vasoconstrictor. Endothelin 1 acts through two types of receptors ETA and ETB [1].
9
9 Cited Publications
Art. -Nr.: HY-P0202A
CAS. Nr.: 394693-38-0
Synonyms: ET-1 (swine, human) TFA
Target:  

Endothelin Receptor

Forschungsgebiete:  

Cardiovascular Disease

Endothelin 1 (swine, human) (ET-1) TFA is a synthetic peptide with the sequence of human and swine Endothelin 1, which is a potent endogenous vasoconstrictor. Endothelin 1 TFA acts through two types of receptors ETA and ETB [1].
7
7 Cited Publications
Art. -Nr.: HY-B1811
CAS. Nr.: 11000-17-2
Synonyms: Arginine vasopressin; Antidiuretic hormone
Vasopressin is a cyclic nonapeptide that is synthesized centrally in the hypothalamus. Vasopressin participates in the hypothalamic-pituitary-adrenal axis, and regulates pituitary corticotropin secretion by potentiating the stimulatory effects of corticotropin releasing factor. Vasopressin also can act as a neurotransmitter, exerting its action by binding to specific G protein-coupled receptors [1] .
4
4 Cited Publications
Art. -Nr.: HY-P1408
CAS. Nr.: 404882-00-4
Target:  

Integrin VEGFR

Forschungsgebiete:  

Cancer

Obtustatin is a non-RGD disintegrin consisting of 41 residues. Obtustatin inhibits the adhesion of α1β1 integrin to type IV Collagen (HY-NP003), blocks α1β1 integrin signaling in endothelial cells, and suppresses FGF2-induced angiogenesis. Obtustatin inhibits tumor progression in mouse models and upregulates VEGF expression in sarcoma-bearing mice. Obtustatin can be used in research related to Lewis lung carcinoma and S-180 sarcoma [1] .
4
4 Cited Publications
Art. -Nr.: HY-P1408A
Target:  

Integrin

Forschungsgebiete:  

Cancer

Obtustatin triacetate is a 41-residue non-RGD disintegrin. Obtustatin triacetate can be isolated from the venom of Vipera lebetina obtusa. Obtustatin triacetate is a potent and selective inhibitor of integrin α1β1 adhesion to type IV collagen. Obtustatin triacetate inhibits angiogenesis and may be used in cancer research [1].
3
3 Cited Publications
Art. -Nr.: HY-P0090
CAS. Nr.: 47931-85-1
Synonyms: Salmon calcitonin
Target:  

CGRP Receptor

Forschungsgebiete:  

Cancer

Calcitonin salmon, a calcium regulating hormone, is a dual-action amylin and calcitonin receptor agonist, could stimulate bone formation and inhibit bone resorption.
3
3 Cited Publications
Art. -Nr.: HY-A0182
CAS. Nr.: 56-59-7
Synonyms: PLV-2
Target:  

Vasopressin Receptor

Forschungsgebiete:  

Cardiovascular Disease

Felypressin (PLV-2) is a non-catecholamine vasoconstrictor and a vasopressin 1 agonist. Felypressin is widely used in dental procedures [1] .
3
3 Cited Publications
Art. -Nr.: HY-A0182A
CAS. Nr.: 914453-97-7
Synonyms: PLV-2 acetate
Target:  

Vasopressin Receptor

Forschungsgebiete:  

Cardiovascular Disease

Felypressin acetate (PLV-2 acetate) is a non-catecholamine vasoconstrictor and a vasopressin 1 agonist. Felypressin acetate is widely used in dental procedures [1] .
2
2 Cited Publications
Art. -Nr.: HY-P2526
CAS. Nr.: 454487-07-1
Target:  

Complement System

Forschungsgebiete:  

Cancer

LyP-1 is a cyclic 9-amino-acids tumor homing peptide and selectively bind to p32 receptors overexpressed in various tumor-associated cells [1].
2
2 Cited Publications
Art. -Nr.: HY-P0004
CAS. Nr.: 50-57-7
Synonyms: Lysine vasopressin; [Lys8]-Vasopressin
Lysipressin (Lysine vasopressin) is antidiuretic hormone that have been found in pigs. Lysipressin activates Oxytocin receptors and adenylate-cyclase. Lysipressin adjusts blood pressure and heart rate. Lysipressin shows antinociceptive activity [1] .
2
2 Cited Publications
Art. -Nr.: HY-P2526A
Target:  

Peptides

Forschungsgebiete:  

Cancer

LyP-1 TFA is a cyclic 9 amino acids tumor homing peptide and selectively bind to p32 receptors overexpressed in various tumor-associated cells [1].
2
2 Cited Publications
Art. -Nr.: HY-17584A
CAS. Nr.: 851199-60-5
Target:  

Guanylate Cyclase

Forschungsgebiete:  

Cancer

Linaclotide acetate is a potent and selective guanylate cyclase C agonist; developed for the treatment of constipation-predominant irritable bowel syndrome (IBS-C) and chronic constipation.
1
1 Cited Publications
Art. -Nr.: HY-P4860
CAS. Nr.: 1802086-30-1
Target:  

Akt Gli JNK PKA

Forschungsgebiete:  

Metabolic Disease

Adropin (34-76) is a secretory domain of Adropin. Adropin (34-76) can inhibit cAMP level and glucose production in hepatocytes, and has a hypoglycemic effect. Adropin (34-76) plays an antifibrotic role by inhibiting the GLI1 signaling pathway [1] .
1
1 Cited Publications
Art. -Nr.: HY-P0204A
Synonyms: Endothelin 3 (Rat,Human) TFA
Forschungsgebiete:  

Neurological Disease

Endothelin-3, human, mouse, rabbit, rat TFA (Endothelin 3 (Rat,Human) TFA) is an adhesion stimulant. Endothelin-3, human, mouse, rabbit, rat TFA stimulates the adhesion of enteric neural crest cells to various ECM components. Endothelin-3, human, mouse, rabbit, rat TFA plays an important role in the maintenance and self-renewal of intestinal progenitor cells, participates in the migration of enteric neural crest cells, and helps maintain a suitable environment for the colonization of enteric neural crest cells. Endothelin-3, human, mouse, rabbit, rat TFA acts synergistically with the β1-integrin signaling pathway during enteric nervous system development. Endothelin-3, human, mouse, rabbit, rat TFA can be used in studies related to distal aganglionosis [1].
1
1 Cited Publications
Art. -Nr.: HY-P0204
CAS. Nr.: 117399-93-6
Synonyms: Endothelin 3 (Rat,Human)
Forschungsgebiete:  

Neurological Disease

Endothelin-3, human, mouse, rabbit, rat (Endothelin 3 (Rat,Human)) is an adhesion stimulant. Endothelin-3, human, mouse, rabbit, rat stimulates the adhesion of enteric neural crest cells to various ECM components. Endothelin-3, human, mouse, rabbit, rat plays an important role in the maintenance and self-renewal of intestinal progenitor cells, participates in the migration of enteric neural crest cells, and helps maintain a suitable environment for the colonization of enteric neural crest cells. Endothelin-3, human, mouse, rabbit, rat acts synergistically with the β1-integrin signaling pathway during enteric nervous system development. Endothelin-3, human, mouse, rabbit, rat can be used in studies related to distal aganglionosis [1].
1
1 Cited Publications
Art. -Nr.: HY-P11143A
Forschungsgebiete:  

Cancer

IL4RPep-1 acetate is an interleukin-4 receptor (IL-4R) binding agent. IL4RPep-1 acetate preferentially binds to cells with high levels of IL-4R expression compared to those with low levels of expression. IL4RPep-1-labeled liposomes containing Doxorubicin (HY-15142A) are internalized by cells more efficiently. IL4RPep-1-labeled liposomes accumulate more effectively within H226 tumors [1].