ABCG2-IN-1
ABCG2-IN-1 (compound K2), a Ko143 analog, is an orally active ABCG2 inhibitor with an IC50 of 0.13 μM. ABCG2-IN-1 has favorable oral pharmacokinetic profiles in mice.
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- CAS No.: 2559759-40-7
- Formule: C26H36N4O4
- Masse moléculaire:468.59
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
IC50: 0.13 μM (ABCG2)[1]
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| A549 | CC50 |
52.2 μM
Compound: K2
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Cytotoxicity against human A549 cells incubated for 72 hrs by MTT assay
Cytotoxicity against human A549 cells incubated for 72 hrs by MTT assay
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[PMID: 37482017] |
Chemical Information
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CAS No. 2559759-40-7
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Masse moléculaire 468.59
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Formule C26H36N4O4
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SMILES
CC(C)C[C@H]1C2=C(C[C@]3([H])N1C([C@@H](NC3=O)CCC(NC(C)(C)C)=O)=O)C4=CC=C(OC)C=C4N2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
ABCG2-IN-1 Related Classifications
HY-155652 Related Classifications
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