3 Results for "

Apatinib

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Apatinib" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-13342S
CAS No.: 2468771-44-8
Purity:  ≥98.0%
Apatinib-d8 (hydrochloride) is the deuterium labeled Apatinib hydrochloride .
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Cat. No.: HY-13342AS
CAS No.: 2468771-43-7
Purity:  92.56%
Synonyms: YN968D1-d8 free base
Apatinib-d8 (free base) is the deuterium labeled Apatinib free base . Apatinib free base (YN968D1 free base) is an orally bioavailable tyrosine kinase inhibitor, which selectively targets VEGFR-2 (IC50=1 nM). Apatinib free base (YN968D1 free base) is an anti-angiogenic drug for the research of advanced or metastatic gastric cancer. Apatinib free base (YN968D1 free base) potently inhibits Ret, c-Kit and c-Src with IC50s of 13, 429 and 530 nM, respectively. It also inhibits cellular phosphorylation of VEGFR-2, c-kit and PDGFRβ .
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Cat. No.: HY-142440S
Apatinib 25-N-oxide-d8 (dihydrochloride) is the deuterium labeled Apatinib 25-N-oxide dihydrochloride .
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