ERG-IN-5
ERG-IN-5 (Compound M1) is a metabolite of ERG-IN-4 (HY-180918), and it is a hERG potassium channel inhibitor with an IC50 of 1.5 μM. ERG-IN-5 is cytotoxic to MTAPdel HCT116 and its CC50 is 28 nM. ERG-IN-5 can be used for the study of colon cancer.
For research use only. We do not sell to patients.
- CAS No.: 3047675-62-4
- Formula: C23H20F3N7O2
- Molecular Weight:483.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 3047675-62-4
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Molecular Weight 483.45
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Formula C23H20F3N7O2
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SMILES
NC1=NC(C=CC(C(N(NC(C2CC2)=O)CC3=NC=C(C(F)(F)F)C=C3)=O)=C4)=C4C5=C1C=NN5C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)