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Cat. No.: HY-159587

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P300-IN-4

P300-IN-4 (compound 6) is a (p300) inhibitor with the IC₅₀ of 12.2 μM.

For research use only. We do not sell to patients.

Formula: C₂₉H₂₈ClIN₄O₅
Molecular Weight:674.91

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

P300-IN-4 Chemical Structure

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

P300-IN-4 (compound 6) is a (p300) inhibitor with the IC₅₀ of 12.2 μM.

All Histone Acetyltransferase Isoforms :

Chemical Information

Molecular Weight 674.91
Formula C₂₉H₂₈ClIN₄O₅
SMILES

CNC(C[C@@H](NC(C1=CC=C2C(N(NC2=C1)CC(C(O)=O)CC3=CC=C(C=C3)Cl)=O)=O)CC4=CC=C(C=C4)I)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (268 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Suo Y, et al. Discovery Small-Molecule p300 Inhibitors Derived from a Newly Developed Indazolone-Focused DNA-Encoded Library. Bioconjug Chem. 2024;35(8):1251-1257. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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