1 Result for "

CCT241736

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "CCT241736" in MCE Product Catalog:

Cat. No.: HY-18161
CAS No.: 1402709-93-6
Target:  

FLT3 Aurora Kinase

Research Areas:  

Cancer

CCT241736 is a potent and orally bioavailable dual FLT3 and Aurora kinase inhibitor, which inhibits Aurora kinases (Aurora-A Kd, 7.5 nM, IC50, 38 nM; Aurora-B Kd, 48 nM), FLT3 kinase (Kd, 6.2 nM), and FLT3 mutants including FLT3-ITD (Kd, 38 nM) and FLT3(D835Y) (Kd, 14 nM).
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