1 Result for "

Darlifarnib

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "Darlifarnib" in MCE Product Catalog:

Cat. No.: HY-172423
CAS No.: 3065226-39-0
Synonyms: KO-2806
Research Areas:  

Cancer

Darlifarnib (KO-2806) is an orally active farnesyl transferase inhibitor. Darlifarnib inhibits the mTORC1 signaling pathway, thereby enhancing the anti-angiogenic properties of tyrosine kinase inhibitors. When used in combination with anti-VEGFR tyrosine kinase inhibitors, Darlifarnib promotes renal cell carcinoma tumor regression and inhibits tumor neovascularization. Darlifarnib sensitizes renal cell carcinoma tumors that progress after anti-VEGFR TKI treatment .
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