1 Result for "

LO-3-63

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "LO-3-63" in MCE Product Catalog:

  • Targets Recommended:
Cat. No.: HY-175187
Target:  

CDK E1/E2/E3 Enzyme

Research Areas:  

Cancer

LO-3-63, a Ribociclib (HY-15777) analog bearing a truncated fumaramide handle, is a PROTAC-like CDK4/6 degrader. LO-3-63 induces CUL4 DCAF16-dependent degradation of CDK4/6 in cells .
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