1 Result for "

PLX51107 (Standard)

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "PLX51107 (Standard)" in MCE Product Catalog:

Cat. No.: HY-111422R
CAS No.: 1627929-55-8
Research Areas:  

Cancer

PLX51107 (Standard) is the analytical standard of PLX51107 (HY-111422). This product is intended for research and analytical applications. PLX51107 is a potent and selective BET inhibitor, with Kds of 1.6, 2.1, 1.7, and 5 nM for BD1 and 5.9, 6.2, 6.1, and 120 nM for BD2 of BRD2, BRD3, BRD4, and BRDT, respectively; PLX51107 also interacts with the bromodomains of CBP and EP300 (Kd, in the 100 nM range).
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