1 Result for "

SeSA-HCPT

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "SeSA-HCPT" in MCE Product Catalog:

Cat. No.: HY-181694
Research Areas:  

Cancer

SeSA-HCPT is an orally active dual-target inhibitor integrating Topo I and HDAC inhibition. SeSA-HCPT induces potent DNA damage, apoptosis, S-phase arrest in prostate cancer cells. SeSA-HCPT inhibits cancer cells proliferation and migration. SeSA-HCPT impairs homologous recombination by suppressing KIF4A-RAD51 signaling. SeSA-HCPT markedly inhibits CRPC tumor growth with minimal systemic toxicity .
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