6 Results for "

Tiprolisant

" in MedChemExpress (MCE) Product Catalog:
Products (6)

6 Results for "Tiprolisant" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-12199
CAS No.: 362665-56-3
Purity:  99.73%
Synonyms: Tiprolisant
Target:  

Histamine Receptor

Research Areas:  

Neurological Disease Endocrinology

Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
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2
2 Cited Publications
Cat. No.: HY-12199B
CAS No.: 903576-44-3
Purity:  99.51%
Synonyms: Ciproxidine; BF 2649
Target:  

Histamine Receptor

Research Areas:  

Neurological Disease Endocrinology

Pitolisant hydrochloride is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
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Cat. No.: HY-12199A
CAS No.: 362665-57-4
Synonyms: Tiprolisant oxalate
Target:  

Histamine Receptor

Research Areas:  

Neurological Disease Endocrinology

Pitolisant oxalate is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
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Cat. No.: HY-12199S1
CAS No.: 2416991-77-8
Synonyms: Tiprolisant-d6
Pitolisant-d6 (Tiprolisant-d6) is deuterium labeled Pitolisant. Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
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Cat. No.: HY-12199S
Synonyms: Tiprolisant-d10
Pitolisant-d10 (Tiprolisant-d10) is deuterium labeled Pitolisant. Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM) .
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Cat. No.: HY-12199R
CAS No.: 362665-56-3
Synonyms: Tiprolisant (Standard)
Pitolisant (Standard) is the analytical standard of Pitolisant. This product is intended for research and analytical applications. Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM).
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