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    PROTAC
  2. Estrogen Receptor/ERR
    PROTAC
  3. ARV-471

ARV-471 

Cat. No.: HY-138642
Handling Instructions

ARV-471 is a best-in-class, orally active estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.

For research use only. We do not sell to patients.

ARV-471 Chemical Structure

ARV-471 Chemical Structure

CAS No. : 2229711-68-4

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5 mg USD 980 Ask For Quote & Lead Time
10 mg USD 1650 Ask For Quote & Lead Time
25 mg USD 3450 Ask For Quote & Lead Time

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Description

ARV-471 is a best-in-class, orally active estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer[1].

IC50 & Target

Estrogen receptor

Clinical Trial
Molecular Weight

723.90

Formula

C₄₅H₄₉N₅O₄

CAS No.
SMILES

O=C([[email protected]@H](N(CC1=C2C=CC(N3CCN(CC4CCN(C5=CC=C([[email protected]]6[[email protected]@H](C7=CC=CC=C7)CCC8=C6C=CC(O)=C8)C=C5)CC4)CC3)=C1)C2=O)CC9)NC9=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

ARV-471ARV471ARV 471Estrogen Receptor/ERRPROTACProteolysis-targeting chimeradegraderbreast cancerInhibitorinhibitorinhibit

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