FMJ-01-042
FMJ-01-042 is a blood-brain barrier-permeable, low-efficacy partial agonist with high affinity (Kᵢ = 4.33 nM) and exceptional subtype selectivity for the dopamine D4 receptor. FMJ-01-042 exhibits good metabolic stability and is suitable for research on neurological and psychiatric disorders.
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- Formule: C24H25N5
- Masse moléculaire:383.49
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
FMJ-01-042 (Compound 18) (90 min) can act as a D4R-mediated β-arrestin recruitment antagonist[1].
FMJ-01-042 exhibited good metabolic stability in rat liver microsomes, with a t1/2 value of 56.77 min[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Masse moléculaire 383.49
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Formule C24H25N5
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SMILES
CC1=CC(N2N=NC(CN3CCN(C4=C5C=CC=CC5=CC=C4)CC3)=C2)=CC=C1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
FMJ-01-042 Related Classifications
HY-181047 Related Classifications
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