VUF-6884
VUF-6884 (Compound 7j) is a histamine receptor (Histamine Receptor) ligand with activity toward human H4R and H1R. Its pEC50 and pKi values against human H4R are 7.70 and 7.55, respectively, while those against human H1R are 8.17 and 8.11, respectively. VUF-6884 competitively binds to the orthosteric binding site of human H4R to displace histamine, and exhibits inverse agonist activity at human H1R.
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- No. CAS: 3455-10-5
- Fòrmula: C18H18ClN3O
- Peso molecular:327.81
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Chemical Information
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No. CAS 3455-10-5
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Peso molecular 327.81
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Fòrmula C18H18ClN3O
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SMILES
ClC1=CC=C2N=C(C=3C=CC=CC3OC2=C1)N4CCN(C)CC4
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
VUF-6884 Related Classifications
HY-124912 Related Classifications
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