5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors

  • J Med Chem. 1998 Jul 2;41(14):2442-4. doi: 10.1021/jm980179c.
J D Albright  1 ,  M F Reich ,  E G Delos Santos ,  J P Dusza ,  F W Sum ,  A M Venkatesan ,  J Coupet ,  P S Chan ,  X Ru ,  H Mazandarani ,  T Bailey
Affiliations
  • 1. Wyeth-Ayerst Research, Pearl River, New York 10965, and Wyeth-Ayerst Research, Princeton, New Jersey 08543-8000, USA.
PMID: 9651149 DOI: 10.1021/jm980179c
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