1. Academic Validation
  2. 5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors

5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors

  • J Med Chem. 1998 Jul 2;41(14):2442-4. doi: 10.1021/jm980179c.
J D Albright 1 M F Reich E G Delos Santos J P Dusza F W Sum A M Venkatesan J Coupet P S Chan X Ru H Mazandarani T Bailey
Affiliations

Affiliation

  • 1 Wyeth-Ayerst Research, Pearl River, New York 10965, and Wyeth-Ayerst Research, Princeton, New Jersey 08543-8000, USA.
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