2 Results for "

1821329-75-2

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "1821329-75-2" in MCE Product Catalog:

Cat. No.: HY-19981B
CAS No.: 1821329-75-2
Synonyms: ARQ-087 dihydrochloride
Target:  

EGFR

Research Areas:  

Cancer

Derazantinib (ARQ-087) dihydrochloride is an ATP competitive and orally activeFGFR inhibitor (IC50s: 1.8 nM for FGFR2, 4.5 nM for FGFR1 and 3). Derazantinib dihydrochloride inhibits FGFR phosphorylation. Derazantinib dihydrochloride inhibits tumor growth in multiple xenograft models .
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3
3 Cited Publications
Cat. No.: HY-19981
CAS No.: 1234356-69-4
Synonyms: ARQ-087
Target:  

FGFR

Research Areas:  

Cancer

Derazantinib (ARQ-087) is an ATP competitive and orally activeFGFR inhibitor (IC50s: 1.8 nM for FGFR2, 4.5 nM for FGFR1 and 3 nM). Derazantinib inhibits FGFR phosphorylation. Derazantinib inhibits tumor growth in multiple xenograft models .
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