2 Results for "

5-HT1A modulator 1

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "5-HT1A modulator 1" in MCE Product Catalog:

Cat. No.: HY-100290
CAS No.: 142477-34-7
Purity:  97.12%
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

5-HT1A modulator 1 displays very high affinities for the 5HT1A, adrenergic α1 and dopamine D2 receptor with IC50s of 2 ±0.3 nM, 10 ± 3 nM and 40 ±9 nM, respectively.
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Cat. No.: HY-10861
CAS No.: 898532-85-9
Purity:  99.75%
Research Areas:  

Neurological Disease

D3/5-HT receptor modulator-1 (compound 5i) is a selective dopamine D3 receptor and 5-HT2A receptor antagonist and a partial 5-HT1A receptor agonist. D3/5-HT receptor modulator-1 shows Ki values of 4.5 nM, 11.9 nM, and 15.3 nM for dopamine D3, 5-HT2A, and 5-HT2A receptors. D3/5-HT receptor modulator-1 has a low affinity for dopamine D2 receptors, 5-HT2C receptors, and hERG channels. D3/5-HT receptor modulator-1 has an atypical antipsychotic profile .
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