2 Results for "

80751-65-1

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "80751-65-1" in MCE Product Catalog:

Cat. No.: HY-10435
CAS No.: 80751-65-1
Synonyms: (±)-SKF-82958; Chloro-APB
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

SKF-82958 ((±)-SKF 82958) is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM) .
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4
4 Cited Publications
Cat. No.: HY-10435A
CAS No.: 74115-01-8
Purity:  99.82%
Synonyms: (±)-SKF-82958 hydrobromide; Chloro-APB hydrobromide
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

SKF-82958 ((±)-SKF 82958) hydrobromide is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM) .
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