1 Result for "

A381393

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "A381393" in MCE Product Catalog:

Cat. No.: HY-116941
CAS No.: 726174-00-1
Purity:  99.92%
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM) .
loading...
    loading...